# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA473104 | 6, NO 711 | IC50 | = | 0.04 | uM | ALA4401737 | 7.40 | nM | Rattus norvegicus | ||
2. | ALA2315957 | 7 | IC50 | = | 0.08 | uM | ALA4401738 | 7.10 | nM | Rattus norvegicus | ||
3. | Tiagabine | tiagabine | IC50 | = | 0.07 | uM | ALA4401737 | 7.16 | nM | Rattus norvegicus | ||
4. | ALA3342191 | 9 | % Inhibition of Control Specific Binding (Mean n=2) | -1.5 | % | ALA4883781 | % | Rattus norvegicus | ||||
5. | A-1155463 | 17, A-1155463 | % Inhibition of Control Specific Binding (Mean n=2) | 17.3 | % | ALA4883781 | % | Rattus norvegicus | ||||
6. | ALA4551344 | EUB0000746 | % Inhibition of Control Specific Binding (Mean n=2) | -10.3 | % | ALA4883700 | % | Rattus norvegicus | ||||
7. | ALA4228713 | 22 | % Inhibition of Control Specific Binding (Mean n=2) | -2.6 | % | ALA4883700 | % | Rattus norvegicus | ||||
8. | ALA2170610 | 60 | % Ctrl | 101 | % | ALA4882341 | Not Active | % | Rattus norvegicus | |||
9. | BI 639667 | 19n | % Ctrl | 89 | % | ALA4882269 | Not Active | % | Rattus norvegicus | |||
10. | ALA3417525 | 69, BI665915 | % Ctrl | 82 | % | ALA4881836 | Not Active | % | Rattus norvegicus | |||
11. | ALA3417525 | 69, BI665915 | % Ctrl | 96 | % | ALA4881738 | Not Active | % | Rattus norvegicus | |||
12. | ALA4066040 | 12 | % Inhibition of Control Specific Binding (Mean n=2) | -15.1 | % | ALA4880558 | % | Rattus norvegicus | ||||
13. | ALA4093612 | 13 | % Inhibition of Control Specific Binding (Mean n=2) | -17.9 | % | ALA4880558 | % | Rattus norvegicus | ||||
14. | ALA4533479 | EUB0000339 | % Inhibition of Control Specific Binding (Mean n=2) | -17.3 | % | ALA4880476 | % | Rattus norvegicus | ||||
15. | A192621 | 38 | % Inhibition of Control Specific Binding (Mean n=2) | -12 | % | ALA4880476 | % | Rattus norvegicus | ||||
16. | ALA1312 | r-T3(4) | IC50 | = | 13 | uM | ALA3417976 | 4.89 | nM | Rattus norvegicus | ||
17. | Tiagabine | tiagabine | IC50 | = | 0.64 | uM | ALA3417976 | 6.19 | nM | Rattus norvegicus | ||
18. | ALA3417707 | 11 | IC50 | = | 2.07 | uM | ALA3417975 | 5.68 | nM | Rattus norvegicus | ||
19. | ALA1191532 | 10 | IC50 | = | 0.08 | uM | ALA3417975 | 7.10 | nM | Rattus norvegicus | ||
20. | ALA1192843 | 9 | IC50 | = | 1.59 | uM | ALA3417975 | 5.80 | nM | Rattus norvegicus |