# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2442940 | 10d | INH | 0 | ALA2446597 | Not Active | % | Homo sapiens | ||||
2. | ALA2424668 | 1 | Ki | = | 5600 | nM | ALA2428810 | 5.25 | nM | Homo sapiens | ||
3. | ALA2017869 | 3 | Ki | = | 8700 | nM | ALA2428810 | 5.06 | nM | Homo sapiens | ||
4. | ALA2419440 | (RS)-14u, 14u, atropisomeric mixture | INH | 0 | ALA2421610 | Active | % | Homo sapiens | ||||
5. | d(CH2)5Tyr(Me)AVP | 9 | IC50 | = | 6.3 | 10'-10M | ALA2394917 | 9.20 | nM | Homo sapiens | ||
6. | d(CH2)5Tyr(Me)AVP | 9 | Ki | = | 3.9 | 10'-10M | ALA2394917 | 9.41 | nM | Homo sapiens | ||
7. | L-368,899 hydrochloride | 5 | Ki | = | 180 | nM | ALA2393935 | 6.75 | nM | Homo sapiens | ||
8. | ALA2391300 | 1 | Ki | = | 620 | nM | ALA2393935 | 6.21 | nM | Homo sapiens | ||
9. | E1R | E1R, 4R,5S-2a | INH | = | 2 | % | ALA2395789 | % | Homo sapiens | |||
10. | d(CH2)5Tyr(Me)AVP | 9 | IC50 | = | 1.9 | nM | ALA2394816 | 8.72 | nM | Homo sapiens | ||
11. | ALA2392692 | 27, GSK2188931B | INH | < | 50 | % | ALA2395674 | % | Homo sapiens | |||
12. | ALA2381116 | 39 | INH | = | 10.9 | % | ALA2384652 | % | Homo sapiens | |||
13. | ALA2087421 | 12d | INH | = | 31 | % | ALA2091436 | % | Homo sapiens | |||
14. | ALA2326501 | 5d | INH | = | 17 | % | ALA2328754 | % | Homo sapiens | |||
15. | ALA377414 | 25 | pKi | = | 6.2 | ALA2039715 | 6.20 | nM | Homo sapiens | |||
16. | ALA2037511 | 69, 69B | pKi | < | 5.2 | ALA2039715 | nM | Homo sapiens | ||||
17. | ALA2024094 | 19a | INH | = | 30.5 | % | ALA2026538 | % | Homo sapiens | |||
18. | ALA2024089 | 13a | INH | 0 | ALA2026538 | Not Determined | % | Homo sapiens | ||||
19. | ALA2024087 | 12a | INH | = | 29.1 | % | ALA2026538 | % | Homo sapiens | |||
20. | ALA2017980 | 13 | Ki | > | 1000 | nM | ALA2019479 | nM | Homo sapiens |