# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | QAV680 | 18 | IC50 | > | 10 | uM | ALA2447515 | nM | Homo sapiens | |||
2. | TG6-129 | SID17503974 | KB | = | 199 | nM | ALA2412172 | nM | Homo sapiens | |||
3. | ALA1361498 | SID17505080 | KB | = | 57 | nM | ALA2412172 | nM | Homo sapiens | |||
4. | ALA1507392 | SID17505097 | KB | = | 360 | nM | ALA2412172 | nM | Homo sapiens | |||
5. | ALA1412254 | SID24782326 | KB | = | 2260 | nM | ALA2412172 | nM | Homo sapiens | |||
6. | ALA1503476 | SID17508450 | KB | = | 1730 | nM | ALA2412172 | nM | Homo sapiens | |||
7. | ALA1410750 | SID26671393 | KB | = | 3250 | nM | ALA2412172 | nM | Homo sapiens | |||
8. | ALA1573791 | SID17504270 | KB | = | 360 | nM | ALA2412172 | nM | Homo sapiens | |||
9. | ALA1550812 | SID17504776 | KB | = | 21000 | nM | ALA2412172 | nM | Homo sapiens | |||
10. | ALA1374570 | SID17508802 | KB | = | 5900 | nM | ALA2412172 | nM | Homo sapiens | |||
11. | Iloprost | Iloprost | IC50 | = | 8.4 | 10'-9M | ALA2394933 | 8.08 | nM | Homo sapiens | ||
12. | Iloprost | Iloprost | Ki | = | 4.8 | 10'-9M | ALA2394933 | 8.32 | nM | Homo sapiens | ||
13. | E1R | E1R, 4R,5S-2a | INH | = | -19 | % | ALA2395804 | % | Homo sapiens | |||
14. | Iloprost | Iloprost | IC50 | = | 13 | nM | ALA2394989 | 7.89 | nM | Homo sapiens | ||
15. | ALA94751 | 4 | IC50 | = | 0.081 | uM | ALA3083992 | 7.09 | nM | Homo sapiens | ||
16. | ALA111612 | 10a | % inhibition | 15 | % | ALA4880289 | Not Active | % | Homo sapiens | |||
17. | ABT-100 | EUB0000289 | % inhibition | < | 10 | % | ALA4880213 | Not Active | % | Homo sapiens | ||
18. | 2-[(1r,4r)-4-{4-[(2R)-4-[(2-ethylphenyl)carbamoyl]-2-methyl-3,4-dihydro-2H-1,4-benzoxazin-7-yl]phenyl}cyclohexyl]acetic acid | 23n | IC50 | = | 1 | uM | ALA3294218 | 6.00 | nM | Homo sapiens | ||
19. | ALA3286704 | 9c, TG7-174 | Kb | = | 85 | uM | ALA3293203 | nM | Homo sapiens | |||
20. | ALA3286702 | 9a, TG7-181 | Kb | > | 10000 | uM | ALA3293203 | nM | Homo sapiens |