# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Harmaline | 4 (Harmaline) | Ki | > | 10 | uM | ALA5235596 | nM | Homo sapiens | |||
2. | Harmalan | 6 | Ki | > | 10 | uM | ALA5235596 | nM | Homo sapiens | |||
3. | 6-Methoxyharmalan | 44 | Ki | > | 10 | uM | ALA5235596 | nM | Homo sapiens | |||
4. | ALA5274306 | 15 | INH | < | 50 | % | ALA5228817 | % | Homo sapiens | |||
5. | ALA5286071 | 20 | IC50 | = | 2470 | nM | ALA5225971 | 5.61 | nM | Homo sapiens | ||
6. | ALA5286066 | 19 | IC50 | = | 2190 | nM | ALA5225971 | 5.66 | nM | Homo sapiens | ||
7. | ALA5278676 | 18 | IC50 | = | 7470 | nM | ALA5225971 | 5.13 | nM | Homo sapiens | ||
8. | ALA5278640 | 17 | IC50 | = | 585 | nM | ALA5225971 | 6.23 | nM | Homo sapiens | ||
9. | ALA5275403 | 16 | IC50 | = | 1970 | nM | ALA5225971 | 5.71 | nM | Homo sapiens | ||
10. | ALA5288633 | 15 | IC50 | = | 4210 | nM | ALA5225971 | 5.38 | nM | Homo sapiens | ||
11. | ALA5273314 | 14 | IC50 | = | 1590 | nM | ALA5225971 | 5.80 | nM | Homo sapiens | ||
12. | ALA5278405 | 13 | IC50 | = | 338 | nM | ALA5225971 | 6.47 | nM | Homo sapiens | ||
13. | ALA5272946 | 12 | IC50 | = | 224 | nM | ALA5225971 | 6.65 | nM | Homo sapiens | ||
14. | ALA2104993 | VORTIOXETINE | Ki | = | 3.7 | nM | ALA5215979 | 8.43 | nM | Homo sapiens | ||
15. | ALA4531220 | EUB0000586 | % of inhibition | = | 21 | % | ALA5214760 | % | Homo sapiens | |||
16. | BAY-474 | EUB0000293 | % of control | = | 32.97 | % | ALA5213240 | % | Homo sapiens | |||
17. | A-1155463 | 17, A-1155463 | Ki | = | 1142.6 | nM | ALA5213800 | 5.94 | nM | Homo sapiens | ||
18. | (S)-ZINC 3573 | EUB0000345 | Ki | = | 3626 | nM | ALA5214387 | 5.44 | nM | Homo sapiens | ||
19. | ALA4594433 | ML-246 | Activity | < | 50 | % | ALA5168967 | % | Homo sapiens | |||
20. | RLX-33 | 33 | INH | < | 50 | % | ALA5167535 | % | Homo sapiens |