| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA204232 | 14 | Ki | = | 0.648 | uM | ALA5214272 | 6.19 | nM | Homo sapiens | ||
| 2. |  ALA372199 | 32 | IC50 | = | 213 | nM | ALA5214012 | 6.67 | nM | Homo sapiens | ||
| 3. |  ALA772 | reserpine(5) | IC50 | = | 15.5 | nM | ALA5209602 | 7.81 | Inhibitor | nM | Homo sapiens | |
| 4. |  Tetrabenazine Racemate | Tetrabenazine | IC50 | = | 19.8 | nM | ALA5209602 | 7.70 | Inhibitor | nM | Homo sapiens | |
| 5. |  ALA5209629 | 137699583 | EC50 | = | 3.56 | uM | ALA5209602 | 5.45 | Substrate | nM | Homo sapiens | |
| 6. |  MAK683 | 78; MAK683 | IC50 | = | 1.8 | uM | ALA5163326 | 5.75 | nM | Homo sapiens | ||
| 7. |  3-Isobutyl-9，10-dimethoxy-2，3，4，6，7，11b-hexahydro-1H-pyrido[2，1-a]isoquinolin-2-ol | [3H]-DHTB | Bmax | = | 41.2 | pmol/mg | ALA4202143 | pmol/mg | Homo sapiens | |||
| 8. | 3-Isobutyl-9，10-dimethoxy-2，3，4，6，7，11b-hexahydro-1H-pyrido[2，1-a]isoquinolin-2-ol | [3H]-DHTB | Activity | 0 | ALA4202138 | Active | Homo sapiens | |||||
| 9. |  ALA4207838 | [3H]-(+)-5b | Bmax | = | 13.5 | pmol/mg | ALA4202143 | pmol/mg | Homo sapiens | |||
| 10. | ALA772 | reserpine(5) | Bmax | = | 0.942 | pmol/mg | ALA4202143 | pmol/mg | Homo sapiens | |||
| 11. |  ALA4213176 | (+/-)-5j | IC50 | = | 142 | nM | ALA4202145 | 6.85 | nM | Homo sapiens | ||
| 12. |  ALA4208250 | (+/-)-5i | IC50 | = | 101 | nM | ALA4202145 | 7.00 | nM | Homo sapiens | ||
| 13. |  ALA4217581 | (+/-)-5h | IC50 | > | 10 | uM | ALA4202145 | nM | Homo sapiens | |||
| 14. |  ALA4212633 | (+/-)-5g | IC50 | > | 10 | uM | ALA4202145 | nM | Homo sapiens | |||
| 15. |  ALA4204449 | (+/-)-5f | IC50 | = | 5800 | nM | ALA4202145 | 5.24 | nM | Homo sapiens | ||
| 16. |  ALA4216117 | (+/-)-5e | IC50 | = | 2700 | nM | ALA4202145 | 5.57 | nM | Homo sapiens | ||
| 17. |  ALA4208779 | (+/-)-5d | IC50 | = | 125 | nM | ALA4202145 | 6.90 | nM | Homo sapiens | ||
| 18. |  ALA4203894 | (+/-)-5c | IC50 | = | 2900 | nM | ALA4202145 | 5.54 | nM | Homo sapiens | ||
| 19. |  ALA4205254 | (+)-5b | IC50 | = | 51.1 | nM | ALA4202145 | 7.29 | nM | Homo sapiens | ||
| 20. | ALA4205254 | (+)-5b | IC50 | = | 16 | nM | ALA4202145 | 7.80 | nM | Homo sapiens |
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