# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3330879 | Scheme 1, R3C1 | Kd | = | 2.08 | nM | ALA3385406 | 8.68 | nM | Homo sapiens | ||
2. | ALA3330880 | page no 492, R1C1 | Kd | = | 0.38 | nM | ALA3385406 | 9.42 | nM | Homo sapiens | ||
3. | ALA437696 | 5 | Activity | = | 67 | mg/dl | ALA868372 | mg/dl | Homo sapiens | |||
4. | ALA203135 | 10 | Activity | = | 12 | mg/dl | ALA868372 | mg/dl | Homo sapiens | |||
5. | ALA206717 | 14 | Activity | = | 146 | mg/dl | ALA868372 | mg/dl | Homo sapiens | |||
6. | ALA11697 | 7 | Activity | = | 23 | mg/dl | ALA868372 | mg/dl | Homo sapiens | |||
7. | Gliquidone | GQ | Activity | = | 162 | mg/dl | ALA868372 | mg/dl | Homo sapiens | |||
8. | Berberine chloride form | 1 | Activity | = | 61 | mg/dl | ALA868372 | mg/dl | Homo sapiens | |||
9. | ALA186684 | fluroethylated repaglinide | IC50 | = | 281 | nM | ALA832318 | 6.55 | nM | Homo sapiens | ||
10. | ALA186684 | fluroethylated repaglinide | Kd | = | 134 | nM | ALA830078 | 6.87 | nM | Homo sapiens | ||
11. | ALA360610 | methoxy-repaglinide | IC50 | = | 163 | nM | ALA832318 | 6.79 | nM | Homo sapiens | ||
12. | ALA360610 | methoxy-repaglinide | Kd | = | 83 | nM | ALA830078 | 7.08 | nM | Homo sapiens | ||
13. | Repaglinide | (S)-6al | IC50 | = | 106 | nM | ALA832318 | 6.97 | nM | Homo sapiens | ||
14. | Repaglinide | (S)-6al | Kd | = | 50 | nM | ALA830078 | 7.30 | nM | Homo sapiens |