# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3087669 | 3h | IC50 | = | 37 | uM | ALA3089256 | 4.43 | nM | Homo sapiens | ||
2. | Citalopram | R,S-citalopram | IC50 | = | 0.01 | uM | ALA3090833 | 8.00 | nM | Homo sapiens | ||
3. | Verapamil | 24 | IC50 | = | 0.01 | uM | ALA3090833 | 8.00 | nM | Homo sapiens | ||
4. | Haloperidol | Haloperidol | IC50 | = | 0.01 | uM | ALA3090833 | 8.00 | nM | Homo sapiens | ||
5. | Fluoxetine | fluoxetine | IC50 | = | 0.01 | uM | ALA3090833 | 8.00 | nM | Homo sapiens | ||
6. | ALA2441200 | 17a | INH | = | 40 | % | ALA2444927 | % | Homo sapiens | |||
7. | ALA2442291 | 11j | INH | = | 11 | % | ALA2446215 | % | Homo sapiens | |||
8. | ALA2443278 | (R)-19 | IC50 | = | 2.3 | uM | ALA2445978 | 5.64 | nM | Homo sapiens | ||
9. | oliceridine | (R)-30, TRV130 | IC50 | = | 6.2 | uM | ALA2445978 | 5.21 | nM | Homo sapiens | ||
10. | ALA2441950 | 2q, More active atropisomer | INH | 0 | ALA2444175 | Not Active | % | Homo sapiens | ||||
11. | ALA2441951 | 2r, More active atropisomer | INH | 0 | ALA2444175 | Not Active | % | Homo sapiens | ||||
12. | ALA2441952 | 2s, BMS-767778, More active atropisomer | INH | 0 | ALA2444175 | Not Active | % | Homo sapiens | ||||
13. | ALA2441953 | 2t, More active atropisomer | INH | 0 | ALA2444175 | Not Active | % | Homo sapiens | ||||
14. | ALA2441954 | 2u, More active atropisomer | INH | 0 | ALA2444175 | Not Active | % | Homo sapiens | ||||
15. | ALA2441955 | 2v, More active atropisomer | INH | 0 | ALA2444175 | Not Active | % | Homo sapiens | ||||
16. | ALA2440456 | 17 | IC50 | = | 27.5 | uM | ALA2447591 | 4.56 | nM | Homo sapiens | ||
17. | ALA2440459 | 20 | IC50 | = | 131 | nM | ALA2447591 | 6.88 | nM | Homo sapiens | ||
18. | ALA2440460 | 21 | IC50 | = | 47.5 | uM | ALA2447591 | 4.32 | nM | Homo sapiens | ||
19. | ALA2440456 | 17 | INH | = | 35 | % | ALA2447583 | % | Homo sapiens | |||
20. | ALA2440459 | 20 | INH | = | 2 | % | ALA2447582 | % | Homo sapiens |