| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  PF-04995274 | 1 | Intrinsic activity | = | 41 | % | ALA2154190 | % | Homo sapiens | |||
| 2. |  PF 04418948 | 15, PF-04418948 | % inhibition | -14 | % | ALA4886939 | Not Active | % | Homo sapiens | |||
| 3. |  ALA4536197 | EUB0000326 | % inhibition | 9 | % | ALA4886749 | Not Active | % | Homo sapiens | |||
| 4. |  A 485 | A-485 | % inhibition | 10 | % | ALA4886544 | Not Active | % | Homo sapiens | |||
| 5. |  ALA3342191 | 9 | % Inhibition of Control Specific Binding (Mean n=2) | -4 | % | ALA4883764 | % | Homo sapiens | ||||
| 6. |  A-1155463 | 17, A-1155463 | % Inhibition of Control Specific Binding (Mean n=2) | 6.7 | % | ALA4883764 | % | Homo sapiens | ||||
| 7. |  ALA4551344 | EUB0000746 | % Inhibition of Control Specific Binding (Mean n=2) | -2 | % | ALA4883683 | % | Homo sapiens | ||||
| 8. |  ALA4228713 | 22 | % Inhibition of Control Specific Binding (Mean n=2) | -1 | % | ALA4883683 | % | Homo sapiens | ||||
| 9. |  ALA3480577 | DDD01251909 | pKi | 5.2 | ALA4880070 | nM | Homo sapiens | |||||
| 10. | ALA3480577 | DDD01251909 | Ki | 6685 | nM | ALA4880070 | nM | Homo sapiens | ||||
| 11. | ALA3480577 | DDD01251909 | % Inhibition | 0 | % | ALA4880070 | Not Active | % | Homo sapiens | |||
| 12. | ALA3480577 | DDD01251909 | Mean fold stimulation | 0.925 | ALA4883508 | Homo sapiens | ||||||
| 13. |  PF-04457845 | 23, PF-04457845 | % inhibition | -8 | % | ALA4883134 | Not Active | % | Homo sapiens | |||
| 14. |  ALA3417525 | 69, BI665915 | % Ctrl | 111 | % | ALA4881675 | Not Active | % | Homo sapiens | |||
| 15. |  ALA4066040 | 12 | % Inhibition of Control Specific Binding (Mean n=2) | 5.3 | % | ALA4880541 | % | Homo sapiens | ||||
| 16. |  ALA4093612 | 13 | % Inhibition of Control Specific Binding (Mean n=2) | 10.2 | % | ALA4880541 | % | Homo sapiens | ||||
| 17. |  ALA4533479 | EUB0000339 | % Inhibition of Control Specific Binding (Mean n=2) | -13.4 | % | ALA4880459 | % | Homo sapiens | ||||
| 18. |  A192621 | 38 | % Inhibition of Control Specific Binding (Mean n=2) | -12.4 | % | ALA4880459 | % | Homo sapiens | ||||
| 19. |  ALA125670 | 9d | IC50 | = | 296 | nM | ALA3222890 | 6.53 | nM | Homo sapiens | ||
| 20. |  ALA124485 | 9b | IC50 | = | 715 | nM | ALA3222890 | 6.15 | nM | Homo sapiens |
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