# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | TP-472 | 1; TP-472 | % of control | = | 48 | % | ALA5214185 | % | Homo sapiens | |||
2. | ALA4518342 | EUB0000744 | Ki | > | 50 | uM | ALA5213974 | nM | Homo sapiens | |||
3. | THPP-1 | THPP-1 | Ki | > | 3300 | uM | ALA5214026 | nM | Homo sapiens | |||
4. | PF 04418948 | 15, PF-04418948 | IC50 | = | 3.5 | uM | ALA5214413 | 5.46 | nM | Homo sapiens | ||
5. | ALA5180169 | 2g | INH | < | 50 | % | ALA5168672 | % | Homo sapiens | |||
6. | ALA5180169 | 2g | IC50 | > | 10000 | nM | ALA5168614 | nM | Homo sapiens | |||
7. | ALA5200705 | 26 | INH | = | 36.2 | % | ALA5164173 | % | Homo sapiens | |||
8. | ALA5203666 | IP2 | INH | = | 84.8 | % | ALA5160398 | % | Homo sapiens | |||
9. | ALA5171560 | 33a | IC50 | > | 10000 | nM | ALA5159514 | nM | Homo sapiens | |||
10. | ALA5175729 | 141 | IC50 | = | 42.6 | uM | ALA5128682 | 4.37 | nM | Homo sapiens | ||
11. | ALA4591417 | 31 | IC50 | > | 100 | uM | ALA4416189 | nM | Homo sapiens | |||
12. | ALA4471352 | 4e | IC50 | > | 10000 | nM | ALA4404711 | nM | Homo sapiens | |||
13. | GSK-2894631A | 1bv | INH | 0 | ALA4402278 | Not Active | % | Homo sapiens | ||||
14. | PDE4 inhibitor 16 | 16 | INH | = | 56.6 | % | ALA4397914 | % | Homo sapiens | |||
15. | BPN14770 | ZATOLMILAST | INH | 0 | ALA4397281 | Not Active | % | Homo sapiens | ||||
16. | Cilostamide | Cilostamide, OPC-3689 | INH | = | 85 | % | ALA4395204 | % | Homo sapiens | |||
17. | Cilostamide | Cilostamide, OPC-3689 | INH | = | 39 | % | ALA4395182 | % | Homo sapiens | |||
18. | Cilostamide | Cilostamide, OPC-3689 | INH | = | 9 | % | ALA4395160 | % | Homo sapiens | |||
19. | ALA4468513 | 3b; DRILS-1765 | INH | = | 1 | % | ALA4395103 | % | Homo sapiens | |||
20. | RK-287107 | 1; RK-287107 | INH | > | 20 | % | ALA4388208 | % | Homo sapiens |