# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Carvedilol | 141 | IC50 | = | 3.59 | uM | ALA3638162 | 5.45 | Original reference for datapoint is pubmed_id: 10440104 | nM | Oryctolagus cuniculus | |
2. | ALA3638049 | 3,7-Diazabicyclo[3.3.1]nonane-3-carboxylic acid, 7-[(2S)-3-(4-cyanophenoxy)-2-hydroxypropyl]-,1,1- dimethylethyl ester (H 345/52) | IC50 | = | 6 | uM | ALA3638122 | 5.22 | Test pulse frequency = 0.1 Hz. Original reference for datapoint is pubmed_id: 11164845 | nM | Oryctolagus cuniculus | |
3. | ALA3638049 | 3,7-Diazabicyclo[3.3.1]nonane-3-carboxylic acid, 7-[(2S)-3-(4-cyanophenoxy)-2-hydroxypropyl]-,1,1- dimethylethyl ester (H 345/52) | IC50 | = | 1.3 | uM | ALA3638121 | 5.89 | Test pulse frequency = 1 Hz. Original reference for datapoint is pubmed_id: 11164845 | nM | Oryctolagus cuniculus | |
4. | (-)-Menthol | (-)-menthol | IC50 | = | 74.6 | uM | ALA3638100 | 4.13 | Original reference for datapoint is pubmed_id: 21081797 | nM | Oryctolagus cuniculus | |
5. | ALA2381008 | 6, BPN-4689 | IC50 | > | 100 | uM | ALA2384387 | nM | Oryctolagus cuniculus | |||
6. | ALA2381009 | 19 | IC50 | = | 13 | uM | ALA2384387 | 4.89 | nM | Oryctolagus cuniculus | ||
7. | ALA2381010 | 24 | IC50 | = | 9.3 | uM | ALA2384387 | 5.03 | nM | Oryctolagus cuniculus | ||
8. | ALA2381011 | 21 | IC50 | = | 3.5 | uM | ALA2384387 | 5.46 | nM | Oryctolagus cuniculus | ||
9. | ALA2381012 | 26 | IC50 | = | 4.7 | uM | ALA2384387 | 5.33 | nM | Oryctolagus cuniculus | ||
10. | ALA2381013 | 30 | IC50 | = | 38 | uM | ALA2384387 | 4.42 | nM | Oryctolagus cuniculus | ||
11. | ALA2381014 | 32 | IC50 | = | 43 | uM | ALA2384387 | 4.37 | nM | Oryctolagus cuniculus | ||
12. | ALA2381015 | 34 | IC50 | = | 15 | uM | ALA2384387 | 4.82 | nM | Oryctolagus cuniculus | ||
13. | ALA2381016 | 37 | IC50 | = | 21 | uM | ALA2384387 | 4.68 | nM | Oryctolagus cuniculus | ||
14. | ALA2381017 | 39 | IC50 | = | 46 | uM | ALA2384387 | 4.34 | nM | Oryctolagus cuniculus | ||
15. | ALA2381018 | 41 | IC50 | = | 3.7 | uM | ALA2384387 | 5.43 | nM | Oryctolagus cuniculus | ||
16. | ALA2381019 | 43 | IC50 | > | 100 | uM | ALA2384387 | nM | Oryctolagus cuniculus | |||
17. | ALA2381020 | 45 | IC50 | > | 100 | uM | ALA2384387 | nM | Oryctolagus cuniculus | |||
18. | ALA2381021 | 47 | IC50 | = | 41 | uM | ALA2384387 | 4.39 | nM | Oryctolagus cuniculus | ||
19. | ALA2381022 | 49 | IC50 | > | 100 | uM | ALA2384387 | nM | Oryctolagus cuniculus | |||
20. | ALA2381023 | 51 | IC50 | > | 100 | uM | ALA2384387 | nM | Oryctolagus cuniculus |