# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5208146 | Rac-5a | Ki | = | 26 | nM | ALA5157652 | 7.58 | nM | Cavia porcellus | ||
2. | Naloxone | naloxone | Ki | = | 7.3 | nM | ALA5157652 | 8.14 | nM | Cavia porcellus | ||
3. | U50488 | 9 | Ki | = | 0.34 | nM | ALA5157652 | 9.47 | nM | Cavia porcellus | ||
4. | ALA5200121 | rac-5b | Ki | = | 23 | nM | ALA5157652 | 7.64 | nM | Cavia porcellus | ||
5. | ALA5190238 | (1R,5S,8S)-5a | Ki | = | 123 | nM | ALA5157652 | 6.91 | nM | Cavia porcellus | ||
6. | ALA5203422 | (1S,5R,8R)-5a | Ki | = | 18 | nM | ALA5157652 | 7.75 | nM | Cavia porcellus | ||
7. | ALA5204863 | (1R,5R,7S)-4b | Ki | = | 531 | nM | ALA5157652 | 6.28 | nM | Cavia porcellus | ||
8. | ALA5178401 | (1S,5S,7R)-4b | Ki | = | 13 | nM | ALA5157652 | 7.89 | nM | Cavia porcellus | ||
9. | ALA5185196 | (1R,5R,7S)-4a | Ki | = | 1750 | nM | ALA5157652 | 5.76 | nM | Cavia porcellus | ||
10. | ALA5173028 | (1S,5S,7R)-4a | Ki | = | 7 | nM | ALA5157652 | 8.15 | nM | Cavia porcellus | ||
11. | ALA5200869 | Exo-4 | Ki | = | 862 | nM | ALA5157652 | 6.06 | nM | Cavia porcellus | ||
12. | ALA5175676 | Endo-4 | Ki | = | 7 | nM | ALA5157652 | 8.15 | nM | Cavia porcellus | ||
13. | 2-(3,4-Dichlorophenyl)-1-[2-(1-pyrrolidinylmethyl)-1-piperidinyl]ethanone | 13 | Ki | = | 0.24 | nM | ALA5157652 | 9.62 | nM | Cavia porcellus | ||
14. | ALA5207267 | Exo-2 | Ki | > | 1000 | nM | ALA5157652 | nM | Cavia porcellus | |||
15. | ALA5196638 | Endo-2 | Ki | = | 73 | nM | ALA5157652 | 7.14 | nM | Cavia porcellus | ||
16. | GR 89696 | S-18, GR-89696 | Ki | = | 0.46 | nM | ALA5157652 | 9.34 | nM | Cavia porcellus | ||
17. | U50488 | 9 | Ki | = | 1.1 | nM | ALA5133631 | 8.96 | nM | Cavia porcellus | ||
18. | ALA5194121 | 8b; AD120 | Ki | > | 10000 | nM | ALA5133631 | nM | Cavia porcellus | |||
19. | ALA5203238 | 8a; AD119 | Ki | > | 10000 | nM | ALA5133631 | nM | Cavia porcellus | |||
20. | ALA5190377 | 7b; AD163 | Ki | > | 10000 | nM | ALA5133631 | nM | Cavia porcellus |