# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Forodesine | 1 | Ki | = | 23 | pM | ALA4369204 | 10.64 | nM | Bos taurus | ||
2. | ALA473922 | 2 | Ki | = | 30 | pM | ALA4369204 | 10.52 | nM | Bos taurus | ||
3. | galidesivir | GALIDESIVIR | Ki | = | 2600000 | pM | ALA4369204 | 5.58 | nM | Bos taurus | ||
4. | ALA4574213 | 4-aza-3-deaza-immH | Ki | = | 422000000 | pM | ALA4369204 | nM | Bos taurus | |||
5. | Forodesine | 1 | t1/2 | = | 4.8 | hr | ALA4369206 | hr | Bos taurus | |||
6. | Forodesine | 1 | Kieq | = | 0.023 | nM | ALA2162052 | nM | Bos taurus | |||
7. | ALA2159649 | 6, aza-DFPP-DG | Kieq | = | 6.8 | nM | ALA2162052 | nM | Bos taurus | |||
8. | ALA236709 | DFPP-DG | Kieq | = | 0.085 | nM | ALA2162052 | nM | Bos taurus | |||
9. | ALA236708 | 1 | Kieq | = | 0.72 | nM | ALA2162052 | nM | Bos taurus | |||
10. | ALA2159650 | DFTHPEP-H | Kieq | = | 63 | nM | ALA2162052 | nM | Bos taurus | |||
11. | ALA1794646 | (S)-PMP-DAP | Kieq | = | 6000 | nM | ALA2162052 | nM | Bos taurus | |||
12. | Hypoxanthine | hypoxanthine | Kieq | = | 2500 | nM | ALA2162052 | nM | Bos taurus | |||
13. | Guanine | guanine | Kieq | = | 4000 | nM | ALA2162052 | nM | Bos taurus | |||
14. | 9-Deazaguanine | 9DG | Kieq | = | 7400 | nM | ALA2162052 | nM | Bos taurus | |||
15. | Hypoxanthine | hypoxanthine | Kd | = | 6.8 | 10'-7M | ALA2162055 | 6.17 | nM | Bos taurus | ||
16. | Hypoxanthine | hypoxanthine | Kd | = | 12.5 | 10'-7M | ALA2162056 | 5.90 | nM | Bos taurus | ||
17. | Guanine | guanine | Kd | = | 1.2 | 10'-7M | ALA2162055 | 6.92 | nM | Bos taurus | ||
18. | Guanine | guanine | Kd | = | 0.16 | uM | ALA2162054 | 6.80 | nM | Bos taurus | ||
19. | 9-Deazaguanine | 9DG | Kd | = | 1.6 | 10'-7M | ALA2162055 | 6.80 | nM | Bos taurus | ||
20. | 9-Deazaguanine | 9DG | Kd | = | 1.7 | 10'-7M | ALA2162054 | 6.77 | nM | Bos taurus |