# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3818718 | 11 | INH | 0 | ALA3821420 | Dose-dependent effect | % | Cavia porcellus | ||||
2. | ALA4784305 | 273 | IC50 | = | 2700 | nM | ALA4732995 | 5.57 | nM | Cavia porcellus | ||
3. | ALA4791620 | 272 | IC50 | = | 1600 | nM | ALA4732995 | 5.80 | nM | Cavia porcellus | ||
4. | ALA64605 | Boc-CCK-4 | IC50 | = | 1800 | nM | ALA4732995 | 5.75 | nM | Cavia porcellus | ||
5. | ALA432015 | 9 | ED50 | > | 10 | uM | ALA4687748 | uM | Cavia porcellus | |||
6. | ALA88239 | 1 | ED50 | = | 0.2 | uM | ALA4687748 | uM | Cavia porcellus | |||
7. | ALA317181 | 5 | ED50 | = | 0.43 | uM | ALA4687748 | uM | Cavia porcellus | |||
8. | ALA2310856 | 16 | IC50 | = | 2.1 | nM | ALA661832 | 8.68 | nM | Cavia porcellus | ||
9. | ALA439591 | 6 | IC50 | = | 4.7 | nM | ALA661832 | 8.33 | nM | Cavia porcellus | ||
10. | ALA353862 | Boc-Trp-Phg-Asp-1Nal-NH2 | Ki | = | 1100 | nM | ALA856757 | 5.96 | nM | Cavia porcellus | ||
11. | ALA412238 | 7 | IC50 | = | 140 | nM | ALA661832 | 6.85 | nM | Cavia porcellus | ||
12. | ALA316949 | 1 | Ratio | = | 1.53 | ALA662499 | Cavia porcellus | |||||
13. | ALA316949 | 1 | IC50 | = | 0.77 | nM | ALA661832 | 9.11 | nM | Cavia porcellus | ||
14. | ALA408286 | 19 | IC50 | = | 900 | nM | ALA661832 | 6.05 | nM | Cavia porcellus | ||
15. | ALA98332 | 18 | IC50 | = | 23 | nM | ALA661832 | 7.64 | nM | Cavia porcellus | ||
16. | ALA436722 | Boc-Trp-Phg-Asp-1Nal-N(CH3)2 | Ki | = | 1000 | nM | ALA856757 | 6.00 | nM | Cavia porcellus | ||
17. | ALA98631 | 11 | IC50 | = | 150 | nM | ALA661832 | 6.82 | nM | Cavia porcellus | ||
18. | ALA414793 | 10 | IC50 | = | 81 | nM | ALA661832 | 7.09 | nM | Cavia porcellus | ||
19. | ALA469973 | 15 | IC50 | 0 | ALA964036 | Not Determined | Cavia porcellus | |||||
20. | ALA482571 | 5 | INH | = | 100 | % | ALA964040 | % | Cavia porcellus |