# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | vaborbactam | 27, RPX7009 | MIC | = | 0.25 | ug ml-1 | ALA3579671 | ug.mL-1 | Enterobacter cloacae | |||
2. | vaborbactam | 27, RPX7009 | MIC | <= | 0.06 | ug ml-1 | ALA3579159 | ug.mL-1 | Enterobacter cloacae | |||
3. | vaborbactam | 27, RPX7009 | MIC | <= | 0.06 | ug ml-1 | ALA3578740 | ug.mL-1 | Enterobacter cloacae | |||
4. | vaborbactam | 27, RPX7009 | MIC | = | 0.25 | ug ml-1 | ALA3579486 | ug.mL-1 | Enterobacter cloacae | |||
5. | ALA495027 | 13 | Ratio | = | 2620 | /s/M | ALA1029918 | /s/M | Enterobacter cloacae | |||
6. | ALA492984 | 17 | Ratio | = | 1690 | /s/M | ALA1029918 | /s/M | Enterobacter cloacae | |||
7. | ALA492985 | 21 | Ratio | = | 40 | /s/M | ALA1029918 | /s/M | Enterobacter cloacae | |||
8. | ALA492983 | 9 | Ratio | = | 158 | /s/M | ALA1029918 | /s/M | Enterobacter cloacae | |||
9. | Cephalothin sodium salt | 24 | Ratio | = | 4.85 | 10'5/s/M | ALA1029918 | 10'5/s/M | Enterobacter cloacae | |||
10. | ALA495199 | 23 | Ratio | = | 6 | 10'4/s/M | ALA1029918 | 10'4/s/M | Enterobacter cloacae | |||
11. | ALA495198 | 15 | Ratio | = | 2620 | /s/M | ALA1029918 | /s/M | Enterobacter cloacae | |||
12. | ALA492592 | 12 | Ratio | = | 25 | /s/M | ALA1029918 | /s/M | Enterobacter cloacae | |||
13. | ALA492985 | 21 | Km | = | 2250 | uM | ALA1029913 | nM | Enterobacter cloacae | |||
14. | ALA492983 | 9 | Km | = | 605 | uM | ALA1029913 | nM | Enterobacter cloacae | |||
15. | Cephalothin sodium salt | 24 | Km | = | 270 | uM | ALA1029913 | nM | Enterobacter cloacae | |||
16. | ALA495199 | 23 | Km | = | 680 | uM | ALA1029913 | nM | Enterobacter cloacae | |||
17. | ALA495198 | 15 | Km | = | 1320 | uM | ALA1029913 | nM | Enterobacter cloacae | |||
18. | ALA492592 | 12 | Km | >= | 400 | uM | ALA1029913 | nM | Enterobacter cloacae | |||
19. | ALA492985 | 21 | Kcat | = | 0.09 | /s | ALA1029913 | /s | Enterobacter cloacae | |||
20. | ALA492983 | 9 | Kcat | = | 0.096 | /s | ALA1029913 | /s | Enterobacter cloacae |