# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5277962 | (N)-mc NBTI | IC50 | = | 30 | nM | ALA5233331 | 7.52 | nM | Homo sapiens | ||
2. | S-(4-Nitrobenzyl)-6-thioinosine | 6n | IC50 | = | 1 | nM | ALA5233331 | 9.00 | nM | Homo sapiens | ||
3. | ALA5270911 | (N)-mc dAdo | IC50 | > | 1000000 | nM | ALA5233328 | nM | Homo sapiens | |||
4. | ALA5285935 | (S)-mc dAdo | IC50 | = | 626000 | nM | ALA5233328 | nM | Homo sapiens | |||
5. | ALA5219347 | 99 | IC50 | = | 0.59 | uM | ALA5216608 | 6.23 | nM | Homo sapiens | ||
6. | ALA1325639 | SID865380 | IC50 | = | 2.38 | uM | ALA5216608 | 5.62 | nM | Homo sapiens | ||
7. | ALA5219061 | 97 | IC50 | = | 18.04 | uM | ALA5216608 | 4.74 | nM | Homo sapiens | ||
8. | ALA5219061 | 97 | IC50 | = | 19.42 | uM | ALA5216606 | 4.71 | nM | Homo sapiens | ||
9. | draflazine | DRAFLAZINE | IC50 | = | 5.3 | nM | ALA5209596 | 8.28 | Inhibitor | nM | Homo sapiens | |
10. | Dipyridamole | Dipyridamole | IC50 | = | 8.1 | nM | ALA5209596 | 8.09 | Inhibitor | nM | Homo sapiens | |
11. | dilazep | Dilazep | IC50 | = | 0.1 | nM | ALA5209596 | 10.00 | Inhibitor | nM | Homo sapiens | |
12. | S-(4-Nitrobenzyl)-6-thioinosine | 6n | IC50 | = | 2.6 | nM | ALA5209596 | 8.59 | Inhibitor | nM | Homo sapiens | |
13. | Adenosine | 2 | EC50 | = | 63 | uM | ALA5209596 | 4.20 | Substrate | nM | Homo sapiens | |
14. | ALA4764619 | 6.3; dFdC-C2-CPP6-3 | IC50 | = | 381 | nM | ALA4699780 | 6.42 | nM | Homo sapiens | ||
15. | ALA4796317 | 6.2; dFdC-C2-CPP6-2 | IC50 | = | 384 | nM | ALA4699780 | 6.42 | nM | Homo sapiens | ||
16. | ALA4800221 | 6.1; dFdC-C2-CPP6-1 | IC50 | = | 380 | nM | ALA4699780 | 6.42 | nM | Homo sapiens | ||
17. | ALA4746302 | 4.3; CPP6-3 | IC50 | > | 1000 | nM | ALA4699780 | nM | Homo sapiens | |||
18. | ALA4778383 | 4.2; CPP6-2 | IC50 | > | 1000 | nM | ALA4699780 | nM | Homo sapiens | |||
19. | ALA4749693 | 4.1; CPP6-1 | IC50 | > | 1000 | nM | ALA4699780 | nM | Homo sapiens | |||
20. | Gemcitabine | Gemzar | IC50 | = | 190 | nM | ALA4699780 | 6.72 | nM | Homo sapiens |