# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Ticagrelor | 17, AZD-6140 | Activity | = | 45.02 | % | ALA5232959 | % | Homo sapiens | |||
2. | ALA5279963 | NSC617595 | Activity | = | 92.8 | % | ALA5232959 | % | Homo sapiens | |||
3. | ALA5288399 | NSC618159 | Activity | = | 29.7 | % | ALA5232959 | % | Homo sapiens | |||
4. | ALA5280208 | NSC380323 | Activity | = | 95 | % | ALA5232959 | % | Homo sapiens | |||
5. | ALA5279963 | NSC617595 | IC50 | = | 4.2 | uM | ALA5232958 | 5.38 | nM | Homo sapiens | ||
6. | ALA5288399 | NSC618159 | IC50 | = | 35 | uM | ALA5232958 | 4.46 | nM | Homo sapiens | ||
7. | ALA5280208 | NSC380323 | IC50 | = | 6.49 | uM | ALA5232958 | 5.19 | nM | Homo sapiens | ||
8. | ALA5288399 | NSC618159 | INH | = | 4.75 | % | ALA5232957 | % | Homo sapiens | |||
9. | ALA5280208 | NSC380323 | INH | = | 22.26 | % | ALA5232957 | % | Homo sapiens | |||
10. | ALA5279963 | NSC617595 | INH | = | 36.96 | % | ALA5232957 | % | Homo sapiens | |||
11. | ALA5288399 | NSC618159 | INH | = | 22.77 | % | ALA5232956 | % | Homo sapiens | |||
12. | ALA5279963 | NSC617595 | INH | = | 38.16 | % | ALA5232956 | % | Homo sapiens | |||
13. | ALA5280208 | NSC380323 | INH | = | 33.65 | % | ALA5232956 | % | Homo sapiens | |||
14. | ALA5288399 | NSC618159 | INH | = | 41.12 | % | ALA5232955 | % | Homo sapiens | |||
15. | ALA5280208 | NSC380323 | INH | = | 57.78 | % | ALA5232955 | % | Homo sapiens | |||
16. | ALA5279963 | NSC617595 | INH | = | 61.84 | % | ALA5232955 | % | Homo sapiens | |||
17. | PPTN | 2 | IC50 | > | 10 | uM | ALA5153188 | nM | Homo sapiens | |||
18. | ALA5206028 | [11C]87 | IC50 | = | 6 | nM | ALA5152323 | 8.22 | nM | Homo sapiens | ||
19. | ALA5179763 | [11C]86; [11C]SMW139 | EC50 | = | 60 | nM | ALA5152322 | 7.22 | nM | Homo sapiens | ||
20. | ALA3623467 | 1d | IC50 | = | 46 | nM | ALA5137305 | 7.34 | nM | Homo sapiens |