# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PF-04971729 | 4, PF-04971729 | IC50 | = | 2 | uM | ALA5247041 | 5.70 | nM | Homo sapiens | ||
2. | ALA429910 | 6, dapagliflozin | IC50 | = | 392 | nM | ALA5247041 | 6.41 | nM | Homo sapiens | ||
3. | Remogliflozin etabonate (GSK189075) | 5b, 189075 | Ki | = | 4520 | nM | ALA5227311 | 5.34 | nM | Homo sapiens | ||
4. | ALA3703920 | BDBM159528 | IC50 | = | 163 | nM | ALA5144624 | 6.79 | nM | Homo sapiens | ||
5. | ALA3654892 | BDBM159551 | IC50 | = | 6283 | nM | ALA5144624 | 5.20 | nM | Homo sapiens | ||
6. | ALA3703804 | BDBM159407 | IC50 | = | 2141 | nM | ALA5144624 | 5.67 | nM | Homo sapiens | ||
7. | ALA3654929 | BDBM159590 | IC50 | = | 9931 | nM | ALA5144624 | 5.00 | nM | Homo sapiens | ||
8. | enavogliflozin | BDBM159529 | IC50 | = | 359 | nM | ALA5144624 | 6.45 | nM | Homo sapiens | ||
9. | ALA3703930 | BDBM159538 | IC50 | = | 4940 | nM | ALA5144624 | 5.31 | nM | Homo sapiens | ||
10. | ALA3703936 | BDBM159544 | IC50 | = | 1368 | nM | ALA5144624 | 5.86 | nM | Homo sapiens | ||
11. | ALA3703800 | BDBM159403 | IC50 | = | 556 | nM | ALA5144624 | 6.25 | nM | Homo sapiens | ||
12. | ALA3703906 | BDBM159514 | IC50 | = | 78.1 | nM | ALA5144624 | 7.11 | nM | Homo sapiens | ||
13. | ALA3703797 | BDBM159400 | IC50 | = | 16.9 | nM | ALA5144624 | 7.77 | nM | Homo sapiens | ||
14. | ALA3703799 | BDBM159402 | IC50 | = | 400 | nM | ALA5144624 | 6.40 | nM | Homo sapiens | ||
15. | ALA3703801 | BDBM159404 | IC50 | = | 34.4 | nM | ALA5144624 | 7.46 | nM | Homo sapiens | ||
16. | ALA3703785 | BDBM159387 | IC50 | = | 15.2 | nM | ALA5144624 | 7.82 | nM | Homo sapiens | ||
17. | ALA3703789 | BDBM159391 | IC50 | = | 37.2 | nM | ALA5144624 | 7.43 | nM | Homo sapiens | ||
18. | ALA5169442 | 48b | EC50 | = | 37 | nM | ALA5129934 | 7.43 | nM | Homo sapiens | ||
19. | KGA-2727 | 33f; KGA-2727 | Ki | = | 97.4 | nM | ALA5129931 | 7.01 | nM | Homo sapiens | ||
20. | ALA5182632 | 29; LP-925219 | IC50 | = | 15.9 | nM | ALA5129926 | 7.80 | nM | Homo sapiens |