# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3895524 | BDBM159600 | IC50 | > | 30000 | nM | ALA3888108 | 374032 | nM | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | ||
2. | Avibactam sodium | AVIBACTAM SODIUM | IC50 | = | 650 | nM | ALA3888108 | 6.19 | 374031 | nM | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |
3. | ALA4111243 | BDBM212441 | IC50 | = | 950 | nM | ALA3888108 | 6.02 | 374030 | nM | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |
4. | ALA3895524 | BDBM159600 | IC50 | > | 30000 | nM | ALA3888108 | 374029 | nM | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | ||
5. | ALA4106650 | BDBM212440 | IC50 | = | 650 | nM | ALA3888108 | 6.19 | 374028 | nM | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |
6. | Piperacillin | Piperacillin | Kcat | = | 2 | /s | ALA1640183 | /s | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |||
7. | Piperacillin | Piperacillin | Kcat/Km | = | 50 | /uM/s | ALA1640187 | /uM/s | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |||
8. | Piperacillin | Piperacillin | Km | = | 100 | uM | ALA1640183 | nM | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |||
9. | penicillin G | Benzylpenicillin | Kcat | = | 15 | /s | ALA1640183 | /s | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |||
10. | penicillin G | Benzylpenicillin | Kcat/Km | = | 430 | /uM/s | ALA1640187 | /uM/s | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |||
11. | penicillin G | Benzylpenicillin | Km | = | 35 | uM | ALA1640183 | nM | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |||
12. | Imipenem | Imipenem | Kcat | = | 0.01 | /s | ALA1640183 | /s | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |||
13. | Imipenem | Imipenem | Kcat/Km | = | 0.5 | /uM/s | ALA1640187 | /uM/s | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |||
14. | Imipenem | Imipenem | Km | = | 20 | uM | ALA1640183 | nM | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |||
15. | Cefepime | 82(Cefepime) | Kcat | = | 0.08 | /s | ALA1640183 | /s | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |||
16. | Cefepime | 82(Cefepime) | Kcat/Km | = | 0.1 | /uM/s | ALA1640187 | /uM/s | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |||
17. | Cefepime | 82(Cefepime) | Km | = | 800 | uM | ALA1640183 | nM | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |||
18. | Cephalothin | Cephalothin | Kcat | = | 44 | /s | ALA1640183 | /s | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |||
19. | Cephalothin | Cephalothin | Kcat/Km | = | 510 | /uM/s | ALA1640187 | /uM/s | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | |||
20. | Cephalothin | Cephalothin | Km | = | 85 | uM | ALA1640183 | nM | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) |