# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4225824 | 6a | IC50 | = | 50 | nM | ALA4357657 | 7.30 | nM | Plasmodium falciparum | ||
2. | ALA4435432 | 69 | IC50 | = | 2000 | nM | ALA4357657 | 5.70 | nM | Plasmodium falciparum | ||
3. | ALA4556003 | 67 | IC50 | = | 100 | nM | ALA4357657 | 7.00 | nM | Plasmodium falciparum | ||
4. | ALA4537622 | 55 | IC50 | = | 104 | nM | ALA4357657 | 6.98 | nM | Plasmodium falciparum | ||
5. | ALA4530972 | 54 | IC50 | = | 113 | nM | ALA4357657 | 6.95 | nM | Plasmodium falciparum | ||
6. | ALA4543535 | 53 | IC50 | = | 1162 | nM | ALA4357657 | 5.93 | nM | Plasmodium falciparum | ||
7. | ALA1230705 | 52 | IC50 | = | 1123 | nM | ALA4357657 | 5.95 | nM | Plasmodium falciparum | ||
8. | ALA4470715 | 51 | IC50 | = | 123 | nM | ALA4357657 | 6.91 | nM | Plasmodium falciparum | ||
9. | ALA1233569 | 50 | IC50 | = | 655 | nM | ALA4357657 | 6.18 | nM | Plasmodium falciparum | ||
10. | ALA4516552 | 39 | IC50 | = | 280 | nM | ALA4357657 | 6.55 | nM | Plasmodium falciparum | ||
11. | ALA176888 | 13 | Ki | = | 0.8 | nM | ALA4357657 | 9.10 | nM | Plasmodium falciparum | ||
12. | ALA4520253 | (S,R)-5b | IC50 | = | 10.3 | uM | ALA4331651 | 4.99 | nM | Plasmodium falciparum | ||
13. | ALA4464784 | (S,R)-5a | IC50 | = | 5.6 | uM | ALA4331651 | 5.25 | nM | Plasmodium falciparum | ||
14. | ALA4449824 | (S,R)-4g | IC50 | = | 0.78 | uM | ALA4331651 | 6.11 | nM | Plasmodium falciparum | ||
15. | ALA4449532 | (S,R)-4c | IC50 | = | 1.1 | uM | ALA4331651 | 5.96 | nM | Plasmodium falciparum | ||
16. | ALA2334376 | 33 | IC50 | = | 3.1 | uM | ALA4331651 | 5.51 | nM | Plasmodium falciparum | ||
17. | ALA4515147 | (S,R)-3h | IC50 | = | 2 | uM | ALA4331651 | 5.70 | nM | Plasmodium falciparum | ||
18. | ALA4454293 | (S,R)-3d | IC50 | = | 2.5 | uM | ALA4331651 | 5.60 | nM | Plasmodium falciparum | ||
19. | ALA4555241 | (S,R)-3b | IC50 | = | 1.8 | uM | ALA4331651 | 5.75 | nM | Plasmodium falciparum | ||
20. | ALA4515257 | (S,R)-3a | IC50 | = | 7.4 | uM | ALA4331651 | 5.13 | nM | Plasmodium falciparum |