# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4535356 | oleoyl-D-Lys; 33 | INH | 0 | ALA4481270 | Not Active | % | Homo sapiens | ||||
2. | ALA4742035 | synthetic Cn2 | INH | 0 | ALA4720268 | Not Active | % | Homo sapiens | ||||
3. | ALA3945969 | BDBM217483 | IC50 | = | 0.39 | uM | ALA4321987 | 6.41 | nM | Homo sapiens | ||
4. | ALA3945969 | BDBM217483 | IC50 | = | 0.003 | uM | ALA4321987 | 8.49 | nM | Homo sapiens | ||
5. | GX 201 | 14; GX-201 | Kd | = | 0.004 | uM | ALA4322019 | 8.46 | nM | Homo sapiens | ||
6. | ALA4471012 | 13; GX-585 | Kd | = | 0.022 | uM | ALA4322019 | 7.66 | nM | Homo sapiens | ||
7. | ALA4458532 | 25 | IC50 | = | 0.044 | uM | ALA4321987 | 7.36 | nM | Homo sapiens | ||
8. | ALA4547737 | 24 | IC50 | = | 0.019 | uM | ALA4321987 | 7.72 | nM | Homo sapiens | ||
9. | saxitoxin | STX | IC50 | = | 0.41 | uM | ALA4321987 | 6.39 | nM | Homo sapiens | ||
10. | Tetrodotoxin | TETRODOTOXIN | IC50 | = | 0.036 | uM | ALA4321987 | 7.44 | nM | Homo sapiens | ||
11. | ALA4454760 | 21; JNJ63955918 | IC50 | = | 0.01 | uM | ALA4321987 | 8.00 | nM | Homo sapiens | ||
12. | ALA3416886 | 1 | IC50 | = | 0.002 | uM | ALA4321987 | 8.68 | nM | Homo sapiens | ||
13. | ALA4588728 | 18; Pn3a, MU-TRTX-Pn3a | IC50 | = | 0.001 | uM | ALA4321987 | 9.05 | nM | Homo sapiens | ||
14. | ALA3318132 | 1 | IC50 | = | 0.001 | uM | ALA4321987 | 9.10 | nM | Homo sapiens | ||
15. | ALA3662190 | BDBM145591 | IC50 | = | 0.001 | uM | ALA4321987 | 9.22 | nM | Homo sapiens | ||
16. | Funapide | FUNAPIDE | IC50 | = | 0.054 | uM | ALA4321987 | 7.27 | nM | Homo sapiens | ||
17. | Raxatrigine | VIXOTRIGINE | IC50 | = | 32 | uM | ALA4321987 | 4.50 | nM | Homo sapiens | ||
18. | PF-05089771 | SI-4, R110C1 | IC50 | = | 0.011 | uM | ALA4321987 | 7.96 | nM | Homo sapiens | ||
19. | ALA3657855 | BDBM145285 | IC50 | = | 0 | uM | ALA4321987 | 9.40 | nM | Homo sapiens | ||
20. | ALA4217988 | 5; PF-06456384 | IC50 | = | 0 | uM | ALA4321987 | 11.00 | nM | Homo sapiens |