# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4577237 | EUB0000549 | Kd | > | 1 | uM | ALA4887050 | Not Active | nM | Homo sapiens | ||
2. | BI-1950 | EUB0000310 | Kd | 9 | nM | ALA4887050 | Active | nM | Homo sapiens | |||
3. | ALA3298198 | 16d | INH | 0 | ALA3379760 | Dose-dependent effect | % | Homo sapiens | ||||
4. | ALA3298197 | 16c | INH | 0 | ALA3379760 | Dose-dependent effect | % | Homo sapiens | ||||
5. | ALA3298196 | 16b | INH | 0 | ALA3379760 | Dose-dependent effect | % | Homo sapiens | ||||
6. | ALA3298195 | 16a | INH | 0 | ALA3379760 | Dose-dependent effect | % | Homo sapiens | ||||
7. | ALA3298661 | 18b | FC | = | 2 | ALA3379764 | Homo sapiens | |||||
8. | ALA3297752 | 18a | FC | = | 3 | ALA3379764 | Homo sapiens | |||||
9. | ALA3298198 | 16d | INH | 0 | ALA3379759 | Active | % | Homo sapiens | ||||
10. | ALA3298197 | 16c | INH | 0 | ALA3379759 | Active | % | Homo sapiens | ||||
11. | ALA3298196 | 16b | INH | 0 | ALA3379759 | Active | % | Homo sapiens | ||||
12. | ALA3298195 | 16a | INH | 0 | ALA3379759 | Active | % | Homo sapiens | ||||
13. | ALA3298198 | 16d | INH | 0 | ALA3379761 | Active | % | Homo sapiens | ||||
14. | ALA3298197 | 16c | INH | 0 | ALA3379761 | Active | % | Homo sapiens | ||||
15. | ALA3298196 | 16b | INH | 0 | ALA3379761 | Active | % | Homo sapiens | ||||
16. | ALA3298195 | 16a | INH | 0 | ALA3379761 | Active | % | Homo sapiens | ||||
17. | ALA3298661 | 18b | IC50 | = | 28 | nM | ALA3379760 | 7.55 | nM | Homo sapiens | ||
18. | ALA3297752 | 18a | IC50 | = | 100 | nM | ALA3379760 | 7.00 | nM | Homo sapiens | ||
19. | ALA3298660 | 17i | IC50 | = | 65 | nM | ALA3379760 | 7.19 | nM | Homo sapiens | ||
20. | ALA3298413 | 17h | IC50 | > | 10000 | nM | ALA3379760 | nM | Homo sapiens |