# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BI-1950 | EUB0000310 | % Ctrl | 73 | % | ALA4887080 | Not Active | % | Rattus norvegicus | |||
2. | BI-1950 | EUB0000310 | % Ctrl | 99 | % | ALA4887079 | Not Active | % | Rattus norvegicus | |||
3. | BI-1950 | EUB0000310 | % Ctrl | 96 | % | ALA4887078 | Not Active | % | Rattus norvegicus | |||
4. | ALA2403318 | BI 207127 | % Ctrl | 148 | % | ALA4885610 | Not Active | % | Rattus norvegicus | |||
5. | ALA4636332 | EUB0001578 | % Ctrl | 127 | % | ALA4885563 | Not Active | % | Rattus norvegicus | |||
6. | BI 99179 | 13, BI-99179 | % Ctrl | 92 | % | ALA4882393 | Not Active | % | Rattus norvegicus | |||
7. | BI 99179 | 13, BI-99179 | % Ctrl | 96 | % | ALA4882392 | Not Active | % | Rattus norvegicus | |||
8. | ALA2170610 | 60 | % Ctrl | 92 | % | ALA4882340 | Not Active | % | Rattus norvegicus | |||
9. | ALA2170610 | 60 | % Ctrl | 89 | % | ALA4882339 | Not Active | % | Rattus norvegicus | |||
10. | BI 639667 | 19n | % Ctrl | 104 | % | ALA4882268 | Not Active | % | Rattus norvegicus | |||
11. | BI 639667 | 19n | % Ctrl | 98 | % | ALA4882267 | Not Active | % | Rattus norvegicus | |||
12. | ALA3417525 | 69, BI665915 | % Ctrl | 115 | % | ALA4881835 | Not Active | % | Rattus norvegicus | |||
13. | ALA3417525 | 69, BI665915 | % Ctrl | 100 | % | ALA4881834 | Not Active | % | Rattus norvegicus | |||
14. | ALA3417525 | 69, BI665915 | % Ctrl | 117 | % | ALA4881705 | Not Active | % | Rattus norvegicus | |||
15. | BI-2545 | 19; BI-2545 | % Ctrl | 136 | % | ALA4881635 | Not Active | % | Rattus norvegicus | |||
16. | ALA911 | 2 | Ki | = | 26.7 | nM | ALA3995200 | 7.57 | nM | Rattus norvegicus | ||
17. | Diazepam | Diazepam | Ki | = | 14 | nM | ALA3995200 | 7.85 | nM | Rattus norvegicus | ||
18. | ALA4081736 | 65 | Ki | = | 7 | nM | ALA3995200 | 8.15 | nM | Rattus norvegicus | ||
19. | ALA4229086 | Table 8, R4C3 | Emax | = | 56 | % | ALA4219577 | % | Rattus norvegicus | |||
20. | ALA4229086 | Table 8, R4C3 | EC50 | = | 15 | uM | ALA4219576 | 4.82 | nM | Rattus norvegicus |