# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3746902 | 46, free amine | IC50 | = | 20.7 | uM | ALA3750551 | 4.68 | nM | Staphylococcus aureus | ||
2. | ceftaroline fosamil | ceftaroline | IC50 | = | 0.034 | ug ml-1 | ALA1667068 | ug.mL-1 | Staphylococcus aureus | |||
3. | ALA1652606 | Ceftobiprole medocaril | IC50 | = | 0.5 | ug ml-1 | ALA1667056 | ug.mL-1 | Staphylococcus aureus | |||
4. | Ceftriaxone | 4 | IC50 | = | 0.1 | ug ml-1 | ALA966188 | ug.mL-1 | Staphylococcus aureus | |||
5. | Ceftazidime (containing approximately 10% sodium carbonate) | CAZ | Activity | 0 | ALA966188 | Not Determined | Staphylococcus aureus | |||||
6. | ceftobiprole | BPR, ceftobiprole | IC50 | = | 0.5 | ug ml-1 | ALA966188 | ug.mL-1 | Staphylococcus aureus | |||
7. | ALA66853 | 15b | IC50 | > | 250 | ug ml-1 | ALA762721 | ug.mL-1 | Staphylococcus aureus | |||
8. | ALA67628 | 11d | IC50 | > | 250 | ug ml-1 | ALA762721 | ug.mL-1 | Staphylococcus aureus | |||
9. | ALA294507 | 23 | IC50 | > | 250 | ug ml-1 | ALA762721 | ug.mL-1 | Staphylococcus aureus | |||
10. | ALA67473 | 22 | IC50 | > | 250 | ug ml-1 | ALA762721 | ug.mL-1 | Staphylococcus aureus | |||
11. | ALA67669 | 26 | IC50 | > | 250 | ug ml-1 | ALA762721 | ug.mL-1 | Staphylococcus aureus | |||
12. | ALA67946 | 25 | IC50 | > | 250 | ug ml-1 | ALA762721 | ug.mL-1 | Staphylococcus aureus | |||
13. | ALA304925 | 19b | IC50 | > | 250 | ug ml-1 | ALA762721 | ug.mL-1 | Staphylococcus aureus | |||
14. | ALA63749 | 24 | IC50 | > | 250 | ug ml-1 | ALA762721 | ug.mL-1 | Staphylococcus aureus | |||
15. | ALA432719 | 20b | IC50 | > | 250 | ug ml-1 | ALA762721 | ug.mL-1 | Staphylococcus aureus | |||
16. | ALA306206 | 12 | IC50 | > | 250 | ug ml-1 | ALA762721 | ug.mL-1 | Staphylococcus aureus | |||
17. | ALA67954 | 19c | IC50 | > | 250 | ug ml-1 | ALA762721 | ug.mL-1 | Staphylococcus aureus | |||
18. | ALA304750 | 21 | IC50 | > | 250 | ug ml-1 | ALA762721 | ug.mL-1 | Staphylococcus aureus | |||
19. | ALA68222 | 11c | IC50 | > | 250 | ug ml-1 | ALA762721 | ug.mL-1 | Staphylococcus aureus | |||
20. | ALA66962 | 11b | IC50 | > | 250 | ug ml-1 | ALA762721 | ug.mL-1 | Staphylococcus aureus |