| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA14 | carbacholine | Activity | = | 60 | % | ALA867989 | % | Torpedo californica | |||
| 2. |  ALA298833 | TPMP | pKapp | = | 5.7 | ALA753098 | Torpedo californica | |||||
| 3. |  ALA111404 | 18 | pKapp | = | 6.01 | ALA753098 | Torpedo californica | |||||
| 4. |  ALA326532 | 7 | pKapp | = | 6.4 | ALA753098 | Torpedo californica | |||||
| 5. |  ALA111324 | 19 | pKapp | = | 5.48 | ALA753098 | Torpedo californica | |||||
| 6. |  ALA1788226 | (R)-2 | EC50 | = | 8 | uM | ALA751480 | 5.10 | nM | Torpedo californica | ||
| 7. | ALA1788226 | (R)-2 | EC50 | = | 31 | uM | ALA751480 | 4.51 | nM | Torpedo californica | ||
| 8. |  ALA1132 | 6 (nornicotine) | Relative potency | = | 0.062 | ALA750384 | Torpedo californica | |||||
| 9. |  Besipirdine | 61 | Activity | 0 | ALA748738 | Not Active | Torpedo californica | |||||
| 10. |  ALA94704 | (Z)-6l | Inhibition | = | 88 | % | ALA747861 | % | Torpedo californica | |||
| 11. |  ALA313865 | (E)-6l | Inhibition | = | 95 | % | ALA747861 | % | Torpedo californica | |||
| 12. |  ALA316780 | (E)-6k | Inhibition | = | 94 | % | ALA747861 | % | Torpedo californica | |||
| 13. |  (±)-Epibatidine | 9 | Ki | = | 100 | pM | ALA748739 | 10.00 | nM | Torpedo californica | ||
| 14. |  Acetylcholine | table I | EC50 | = | 5 | uM | ALA750566 | 5.30 | nM | Torpedo californica | ||
| 15. |  ALA335712 | 14 | EC50 | = | 2000 | uM | ALA750566 | nM | Torpedo californica | |||
| 16. |  3-Methyl-5-(1-methyl-2-pyrrolidinyl)isoxazole | 4a | EC50 | = | 411 | uM | ALA750566 | nM | Torpedo californica | |||
| 17. |  ALA328754 | isoquinoline | Kd2 | = | 51.6 | uM | ALA753095 | uM | Torpedo californica | |||
| 18. | ALA328754 | isoquinoline | Kd1 | = | 3.1 | uM | ALA752925 | uM | Torpedo californica | |||
| 19. | ALA328754 | isoquinoline | Bmax | = | 0.31 | uM | ALA752923 | uM | Torpedo californica | |||
| 20. | ALA328754 | isoquinoline | Kd2 | = | 49 | uM | ALA752927 | uM | Torpedo californica |
The page will load shortly, Thanks for your patience!