Activities

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Activities

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#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Assay Description	Assay	Assay Organism
1.	ALA3741992	15	INH	<	30	%	ALA3744784		%	Homo sapiens
2.	ALA3622360	21c	INH	=	-22	%	ALA3624145		%	Homo sapiens
3.	MK-0974	38, MK-0974	pA2	=	8.43		ALA3370794	8.43	nM	Homo sapiens
4.	Olcegepant	BIBN 4096 BS	pA2	=	10.4		ALA3370794	10.40	nM	Homo sapiens
5.	Olcegepant	BIBN 4096 BS	pA2	=	10.1		ALA3370793	10.10	nM	Homo sapiens
6.	MK-3207	3, MK-3207	t1/2	=	59	min	ALA3370562		hr	Homo sapiens
7.	MK-0974	38, MK-0974	t1/2	=	1.3	min	ALA3370562		hr	Homo sapiens
8.	MK-0974	38, MK-0974	K	=	0.51	/min	ALA3370561		/min	Homo sapiens
9.	MK-0974	38, MK-0974	Kd	=	1.9	nM	ALA3370560	8.72	nM	Homo sapiens
10.	MK-0974	38, MK-0974	IC50	=	11	nM	ALA3370558	7.96	nM	Homo sapiens
11.	MK-0974	38, MK-0974	IC50	=	2.2	nM	ALA3370557	8.66	nM	Homo sapiens
12.	ALA3334623	4	IC50	=	44	nM	ALA3370549	7.36	nM	Homo sapiens
13.	4-(2-Oxo-1,2,4,5-tetrahydro-3H-1,3-benzodiazepine-3-yl)piperidine-1-carboxylic acid (R)-alpha-((4-morpholinopiperidino)carbonyl)-3,5-dimethyl-4-hydroxyphenethyl ester	5, BI 44370	Ki	=	0.3	nM	ALA3370549	9.52	nM	Homo sapiens
14.	Olcegepant	BIBN 4096 BS	IC50	=	0.03	nM	ALA3370549	10.52	nM	Homo sapiens
15.	Olcegepant	BIBN 4096 BS	Ki	=	0.014	nM	ALA3370550	10.85	nM	Homo sapiens
16.	ALA196582	3	IC50	=	17000	nM	ALA3370549	4.77	nM	Homo sapiens
17.	MK-0974	38, MK-0974	Ki	=	0.77	nM	ALA3370550	9.11	nM	Homo sapiens
18.	ALA4202767	56	Activity	<=	25	%	ALA4187086		%	Homo sapiens
19.	Olcegepant	BIBN 4096 BS	Ratio Ki	=	150		ALA3292880			Homo sapiens
20.	ALA3288290	8	EC50	=	100	nM	ALA3292879	7.00	nM	Homo sapiens