# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5271559 | 3 | IC50 | > | 2500 | nM | ALA5252501 | nM | Homo sapiens | |||
2. | ALA3823844 | 12 | IC50 | = | 35 | nM | ALA5246064 | 7.46 | nM | Homo sapiens | ||
3. | ALA3699142 | BDBM142744 | IC50 | = | 25 | nM | ALA5246058 | 7.60 | nM | Homo sapiens | ||
4. | JNJ-7706621 | 3b | IC50 | = | 11 | nM | ALA5246051 | 7.96 | nM | Homo sapiens | ||
5. | ALA5278077 | 4; AJI-100 | IC50 | = | 5.4 | nM | ALA5246051 | 8.27 | nM | Homo sapiens | ||
6. | ALA2170414 | 9m | IC50 | = | 5.7 | nM | ALA5246051 | 8.24 | nM | Homo sapiens | ||
7. | ALA5287203 | 12b | INH | < | 40 | % | ALA5244053 | % | Homo sapiens | |||
8. | ALA5267815 | 12a | INH | < | 40 | % | ALA5244053 | % | Homo sapiens | |||
9. | ALA5285244 | 11f | INH | < | 40 | % | ALA5244053 | % | Homo sapiens | |||
10. | ALA5274296 | 11d | INH | < | 40 | % | ALA5244053 | % | Homo sapiens | |||
11. | Alisertib (MLN8237) | 9, MLN-8237 | INH | 0 | ALA5243985 | Active | % | Homo sapiens | ||||
12. | ALA5288971 | 9a | Activity | = | 115 | % | ALA5243966 | % | Homo sapiens | |||
13. | ALA5288971 | 9a | Activity | = | 109 | % | ALA5243965 | % | Homo sapiens | |||
14. | ALA5288971 | 9a | Activity | = | 106 | % | ALA5243964 | % | Homo sapiens | |||
15. | ALA5289096 | h6 | Activity | = | 100 | % | ALA5243963 | % | Homo sapiens | |||
16. | ALA5289096 | h6 | Activity | = | 100 | % | ALA5243962 | % | Homo sapiens | |||
17. | ALA5289096 | h6 | Activity | = | 100 | % | ALA5243961 | % | Homo sapiens | |||
18. | ALA5286283 | 1 | IC50 | = | 35 | nM | ALA5241183 | 7.46 | nM | Homo sapiens | ||
19. | ALA5288241 | B2 | INH | = | 68 | % | ALA5238239 | % | Homo sapiens | |||
20. | ALA5278315 | 18; JB170 | Emax | = | 300 | nM | ALA5238035 | nM | Homo sapiens |