# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2425654 | 3 | INH | = | 100 | % | ALA2429675 | % | Homo sapiens | |||
2. | ALA2425652 | 4 | INH | = | 91 | % | ALA2429675 | % | Homo sapiens | |||
3. | ALA2425649 | 8 | INH | = | 100 | % | ALA2429675 | % | Homo sapiens | |||
4. | ALA2425645 | 11 | INH | = | 100 | % | ALA2429675 | % | Homo sapiens | |||
5. | ALA2425644 | 13 | INH | = | 100 | % | ALA2429675 | % | Homo sapiens | |||
6. | ALA2425646 | 12 | INH | = | 91 | % | ALA2429675 | % | Homo sapiens | |||
7. | ALA1898211 | SID124360154 | Activity | < | 30 | % | ALA2394177 | % | Homo sapiens | |||
8. | (1S,2S,3R,4R)-3-[[5-chloro-2-[(1-ethyl-6-methoxy-2-oxo-4,5-dihydro-3H-1-benzazepin-7-yl)amino]pyrimidin-4-yl]amino]bicyclo[2.2.1]hept-5-ene-2-carboxamide | 15 | INH | < | 50 | % | ALA2046179 | % | Homo sapiens | |||
9. | (1S,2S,3R,4R)-3-[[5-chloro-2-[(1-ethyl-6-methoxy-2-oxo-4,5-dihydro-3H-1-benzazepin-7-yl)amino]pyrimidin-4-yl]amino]bicyclo[2.2.1]hept-5-ene-2-carboxamide | 15 | INH | = | 91 | % | ALA2046178 | % | Homo sapiens | |||
10. | ALA2029438 | 2s | Activity | 0 | ALA2033665 | Active | Homo sapiens | |||||
11. | ALA5306285 | EUB0002235 | delta Tm Staurosporine positive control | = | 8.714 | ALA5304823 | Homo sapiens | |||||
12. | ALA5306285 | EUB0002235 | delta Tm | = | -0.037 | ALA5304823 | Not Active | Homo sapiens | ||||
13. | ALA5308262 | EUB0002234 | delta Tm Staurosporine positive control | = | 8.714 | ALA5304719 | Homo sapiens | |||||
14. | ALA5308262 | EUB0002234 | delta Tm | = | -0.217 | ALA5304719 | Not Active | Homo sapiens | ||||
15. | ALA5308250 | EUB0002186 | delta Tm Staurosporine positive control | = | 9.892 | ALA5304620 | Homo sapiens | |||||
16. | ALA5308250 | EUB0002186 | delta Tm | = | -1.009 | ALA5304620 | Not Active | Homo sapiens | ||||
17. | ALA5306577 | EUB0002354 | delta Tm Staurosporine positive control | = | 9.892 | ALA5304521 | Homo sapiens | |||||
18. | ALA5306577 | EUB0002354 | delta Tm | = | -1.15 | ALA5304521 | Not Active | Homo sapiens | ||||
19. | ALA4080797 | 35 | Activity | = | 100 | % | ALA4055087 | % | Homo sapiens | |||
20. | ALA4096145 | 2 | Activity | = | 91 | % | ALA4055087 | % | Homo sapiens |