# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BI-409306 | BI-409306 | IC50 | = | 65 | nM | ALA5233303 | 7.19 | nM | Homo sapiens | ||
2. | ALA5281523 | 183, AG-690/40135604 | IC50 | = | 8 | uM | ALA5226664 | 5.10 | nM | Homo sapiens | ||
3. | ALA5267538 | 182 | IC50 | = | 0.025 | uM | ALA5226664 | 7.60 | nM | Homo sapiens | ||
4. | ALA5277578 | 181 | IC50 | = | 0.056 | uM | ALA5226664 | 7.25 | nM | Homo sapiens | ||
5. | ALA5283359 | 184 | IC50 | = | 2.1 | uM | ALA5226664 | 5.68 | nM | Homo sapiens | ||
6. | ALA4547969 | 90 | IC50 | = | 0.034 | uM | ALA5226663 | nM | Homo sapiens | |||
7. | ALA4644938 | (R)-C33 | IC50 | = | 0.056 | uM | ALA5226627 | 7.25 | nM | Homo sapiens | ||
8. | ALA5285855 | 10-(S) | IC50 | = | 0.011 | uM | ALA5226627 | 7.96 | nM | Homo sapiens | ||
9. | ALA4642517 | C33 | IC50 | = | 0.016 | uM | ALA5226627 | 7.80 | nM | Homo sapiens | ||
10. | ALA4649493 | 2 | IC50 | > | 10 | uM | ALA5226627 | nM | Homo sapiens | |||
11. | ALA5219813 | 135 | IC50 | = | 17 | nM | ALA5216436 | 7.77 | nM | Homo sapiens | ||
12. | ALA5221005 | 134 | IC50 | = | 14 | nM | ALA5216436 | 7.85 | nM | Homo sapiens | ||
13. | ALA4518342 | EUB0000744 | Ki | > | 54.55 | uM | ALA5213981 | nM | Homo sapiens | |||
14. | THPP-1 | THPP-1 | Ki | > | 50 | uM | ALA5214033 | nM | Homo sapiens | |||
15. | ALA5180169 | 2g | INH | < | 50 | % | ALA5168674 | % | Homo sapiens | |||
16. | ALA5180169 | 2g | IC50 | > | 10000 | nM | ALA5168619 | nM | Homo sapiens | |||
17. | ALA5171560 | 33a | IC50 | > | 10000 | nM | ALA5159516 | nM | Homo sapiens | |||
18. | ALA5198935 | 30-distomer | IC50 | > | 10 | uM | ALA5154145 | nM | Homo sapiens | |||
19. | ALA5205373 | 13A | IC50 | = | 3 | nM | ALA5154145 | 8.52 | nM | Homo sapiens | ||
20. | ALA5207692 | 36-rac | IC50 | = | 13 | nM | ALA5154145 | 7.89 | nM | Homo sapiens |