# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5276374 | (S)-20a; BGB-8035 | IC50 | > | 200 | uM | ALA5251958 | nM | Homo sapiens | |||
2. | Isavuconazole | isavuconazole | Activity | = | 42 | % | ALA5247000 | % | Homo sapiens | |||
3. | ALA5289695 | 16 | IC50 | > | 15 | uM | ALA5225640 | nM | Homo sapiens | |||
4. | ALA5290029 | 33 | IC50 | > | 40000 | uM | ALA5224659 | nM | Homo sapiens | |||
5. | ALA5279298 | 12l | Activity | 0 | ALA5223914 | Not Active | Homo sapiens | |||||
6. | ALA5220884 | 49 | INH | < | 10 | % | ALA5218071 | % | Homo sapiens | |||
7. | ALA5219762 | Cpd 16 | INH | 0 | ALA5217002 | Active | % | Homo sapiens | ||||
8. | ALA5220410 | Cpd 14 | INH | 0 | ALA5217002 | Active | % | Homo sapiens | ||||
9. | ALA5220856 | Cpd 23; S-d4 | INH | 0 | ALA5217001 | Active | % | Homo sapiens | ||||
10. | ALA5219205 | Cpd 24; R-d4 | INH | 0 | ALA5217001 | Active | % | Homo sapiens | ||||
11. | ALA251643 | 019, bupropion (R) | INH | 0 | ALA5217000 | Active | % | Homo sapiens | ||||
12. | ALA5219205 | Cpd 24; R-d4 | INH | 0 | ALA5217000 | Active | % | Homo sapiens | ||||
13. | ALA5219762 | Cpd 16 | FC | = | 5 | ALA5216999 | Homo sapiens | |||||
14. | ALA5220856 | Cpd 23; S-d4 | FC | = | 5 | ALA5216999 | Homo sapiens | |||||
15. | ALA5220410 | Cpd 14 | FC | = | 15 | ALA5216998 | Homo sapiens | |||||
16. | ALA5219205 | Cpd 24; R-d4 | FC | = | 15 | ALA5216998 | Homo sapiens | |||||
17. | ALA5219762 | Cpd 16 | CL | = | 5.28 | nL/pmol/min | ALA5216997 | nL/pmol/min | Homo sapiens | |||
18. | ALA5220410 | Cpd 14 | CL | = | 0.88 | nL/pmol/min | ALA5216997 | nL/pmol/min | Homo sapiens | |||
19. | ALA5220856 | Cpd 23; S-d4 | CL | = | 25.6 | nL/pmol/min | ALA5216996 | nL/pmol/min | Homo sapiens | |||
20. | ALA5219205 | Cpd 24; R-d4 | CL | = | 13.7 | nL/pmol/min | ALA5216996 | nL/pmol/min | Homo sapiens |