# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | 4-(4-Fluorobenzyl)-8-(1H-pyrrolo[2,3-b]pyridin-5-yl)-3,4-dihydrobenzo[f][1,4]oxazepin-5(2H)-one | 21k | IC50 | = | 3.657 | uM | ALA5156973 | 5.44 | nM | Homo sapiens | ||
2. | ALA4457828 | 7; S-49164 | Time | = | 0.2 | s | ALA4428668 | hr | Homo sapiens | |||
3. | ALA4522750 | 6; S-49513 | Time | = | 0.7 | s | ALA4428668 | hr | Homo sapiens | |||
4. | ALA4534484 | 5 | Time | = | 6.3 | s | ALA4428668 | hr | Homo sapiens | |||
5. | GKA 50 | GKA50 | Time | = | 1.6 | s | ALA4428668 | hr | Homo sapiens | |||
6. | ALA4483049 | 3 | Time | = | 2.7 | s | ALA4428668 | hr | Homo sapiens | |||
7. | ALA1783734 | 2 | Time | = | 8.3 | s | ALA4428668 | hr | Homo sapiens | |||
8. | ALA4457828 | 7; S-49164 | K | = | 5.6 | /s | ALA4428667 | /s | Homo sapiens | |||
9. | ALA4522750 | 6; S-49513 | K | = | 1.4 | /s | ALA4428667 | /s | Homo sapiens | |||
10. | ALA4534484 | 5 | K | = | 0.16 | /s | ALA4428667 | /s | Homo sapiens | |||
11. | GKA 50 | GKA50 | K | = | 0.61 | /s | ALA4428667 | /s | Homo sapiens | |||
12. | ALA4483049 | 3 | K | = | 0.37 | /s | ALA4428667 | /s | Homo sapiens | |||
13. | ALA1783734 | 2 | K | = | 0.12 | /s | ALA4428667 | /s | Homo sapiens | |||
14. | ALA4457828 | 7; S-49164 | K | = | 1.3 | 10'6/s/M | ALA4428665 | 10'6/s/M | Homo sapiens | |||
15. | ALA4522750 | 6; S-49513 | K | = | 0.7 | 10'6/s/M | ALA4428665 | 10'6/s/M | Homo sapiens | |||
16. | ALA4534484 | 5 | K | = | 0.2 | 10'6/s/M | ALA4428665 | 10'6/s/M | Homo sapiens | |||
17. | GKA 50 | GKA50 | K | = | 0.2 | 10'6/s/M | ALA4428665 | 10'6/s/M | Homo sapiens | |||
18. | ALA4483049 | 3 | K | = | 0.9 | 10'6/s/M | ALA4428665 | 10'6/s/M | Homo sapiens | |||
19. | ALA1783734 | 2 | K | = | 0.1 | 10'6/s/M | ALA4428665 | 10'6/s/M | Homo sapiens | |||
20. | ALA4534484 | 5 | Activity | = | 60 | % | ALA4428666 | % | Homo sapiens |