# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3686863 | BDBM142234 | IC50 | = | 12 | nM | ALA3795734 | 7.92 | nM | Rattus norvegicus | ||
2. | Grapiprant (CJ-023,423) | GRAPIPRANT | pA2 | = | 8.19 | ALA3997103 | 8.19 | nM | Rattus norvegicus | |||
3. | ALA4099851 | 4j; AAT-008 | pA2 | = | 8.34 | ALA3997103 | 8.34 | nM | Rattus norvegicus | |||
4. | Grapiprant (CJ-023,423) | GRAPIPRANT | Ki | = | 20 | nM | ALA3997104 | 7.70 | nM | Rattus norvegicus | ||
5. | ALA4099851 | 4j; AAT-008 | Ki | = | 6.1 | nM | ALA3997104 | 8.21 | nM | Rattus norvegicus | ||
6. | ALA2037292 | 4q | EC50 | = | 4.9 | nM | ALA2038102 | 8.31 | nM | Rattus norvegicus | ||
7. | ALA2037291 | 4p | EC50 | = | 7.7 | nM | ALA2038102 | 8.11 | nM | Rattus norvegicus | ||
8. | ALA2037290 | 4o | EC50 | = | 28 | nM | ALA2038102 | 7.55 | nM | Rattus norvegicus | ||
9. | ALA2037289 | 4n | EC50 | = | 1.6 | nM | ALA2038102 | 8.80 | nM | Rattus norvegicus | ||
10. | ALA2036326 | 4m | EC50 | = | 8.8 | nM | ALA2038102 | 8.06 | nM | Rattus norvegicus | ||
11. | ALA2036325 | 4l | EC50 | = | 9.7 | nM | ALA2038102 | 8.01 | nM | Rattus norvegicus | ||
12. | ALA2036324 | 4k | EC50 | = | 13 | nM | ALA2038102 | 7.89 | nM | Rattus norvegicus | ||
13. | ALA2036323 | 4j | EC50 | = | 2.2 | nM | ALA2038102 | 8.66 | nM | Rattus norvegicus | ||
14. | ALA2036322 | 4i | EC50 | = | 5.3 | nM | ALA2038102 | 8.28 | nM | Rattus norvegicus | ||
15. | ALA1957437 | 18 | EC50 | = | 480 | nM | ALA2038102 | 6.32 | nM | Rattus norvegicus | ||
16. | ALA2036321 | 4g | EC50 | = | 21 | nM | ALA2038102 | 7.68 | nM | Rattus norvegicus | ||
17. | ALA2036320 | 4f | EC50 | = | 160 | nM | ALA2038102 | 6.80 | nM | Rattus norvegicus | ||
18. | ALA2036319 | 4e | EC50 | = | 15 | nM | ALA2038102 | 7.82 | nM | Rattus norvegicus | ||
19. | ALA1957436 | 17 | EC50 | = | 27 | nM | ALA2038102 | 7.57 | nM | Rattus norvegicus | ||
20. | ALA2036318 | 4c | EC50 | = | 15 | nM | ALA2038102 | 7.82 | nM | Rattus norvegicus |