# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA492654 | rac-4 | IC50 | = | 0.41 | nM | ALA1023823 | 9.39 | nM | Oryctolagus cuniculus | ||
2. | ALA523836 | (R,R)-5 | IC50 | = | 4.5 | nM | ALA1023823 | 8.35 | nM | Oryctolagus cuniculus | ||
3. | ALA492655 | (R,R)-6 | IC50 | = | 18.6 | nM | ALA1023823 | 7.73 | nM | Oryctolagus cuniculus | ||
4. | ALA495113 | (R,R)-30 | IC50 | = | 9.3 | nM | ALA1023823 | 8.03 | nM | Oryctolagus cuniculus | ||
5. | ALA523352 | (R,R)-31 | IC50 | = | 6.1 | nM | ALA1023823 | 8.21 | nM | Oryctolagus cuniculus | ||
6. | ALA201782 | (-)-34a | IC50 | = | 0.32 | nM | ALA1023823 | 9.49 | nM | Oryctolagus cuniculus | ||
7. | relacatib | 10 | IC50 | = | 0.5 | nM | ALA945089 | 9.30 | nM | Oryctolagus cuniculus | ||
8. | Odanacatib (MK-0822) | 24, odanacatib | IC50 | = | 1 | nM | ALA945089 | 9.00 | nM | Oryctolagus cuniculus | ||
9. | balicatib | 18p | IC50 | = | 2.7 | nM | ALA945089 | 8.57 | nM | Oryctolagus cuniculus | ||
10. | L-873724 | 22 | IC50 | = | 0.8 | nM | ALA945089 | 9.10 | nM | Oryctolagus cuniculus | ||
11. | ALA201914 | rac-34a | IC50 | = | 0.5 | nM | ALA886077 | 9.30 | nM | Oryctolagus cuniculus | ||
12. | ALA245759 | 2, racemic | IC50 | = | 2 | nM | ALA886077 | 8.70 | nM | Oryctolagus cuniculus | ||
13. | ALA247587 | 3, racemic | IC50 | = | 1 | nM | ALA886077 | 9.00 | nM | Oryctolagus cuniculus | ||
14. | ALA391959 | 4, racemic | IC50 | = | 1 | nM | ALA886077 | 9.00 | nM | Oryctolagus cuniculus | ||
15. | ALA247783 | 5, racemic | IC50 | = | 5 | nM | ALA886077 | 8.30 | nM | Oryctolagus cuniculus | ||
16. | ALA245381 | 6, racemic | IC50 | = | 6 | nM | ALA886077 | 8.22 | nM | Oryctolagus cuniculus | ||
17. | ALA395697 | 7, racemic | IC50 | = | 5 | nM | ALA886077 | 8.30 | nM | Oryctolagus cuniculus | ||
18. | ALA245579 | 8, racemic | IC50 | = | 9 | nM | ALA886077 | 8.05 | nM | Oryctolagus cuniculus | ||
19. | ALA245580 | 9, racemic | IC50 | = | 0.1 | nM | ALA886077 | 10.00 | nM | Oryctolagus cuniculus | ||
20. | ALA395698 | 10, racemic | IC50 | = | 0.4 | nM | ALA886077 | 9.40 | nM | Oryctolagus cuniculus |