# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | NU7441 (KU-57788) | 22g | IC50 | > | 10 | uM | ALA2423430 | nM | Homo sapiens | |||
2. | KU-0060648 | 6, KU-0060648 | IC50 | > | 10 | uM | ALA2423430 | nM | Homo sapiens | |||
3. | LY294002 | 2 (LY-294002) | IC50 | > | 10 | uM | ALA2423430 | nM | Homo sapiens | |||
4. | BYL719 | 8, NVP-BYL719 | IC50 | > | 10 | uM | ALA2400704 | nM | Homo sapiens | |||
5. | AZ20 | 6, AZ20 | IC50 | > | 30 | uM | ALA2330563 | nM | Homo sapiens | |||
6. | ALA5201686 | 10f | Activity | > | 75 | % | ALA5158119 | % | Homo sapiens | |||
7. | BAY-091 | EUB0001564 | % inhibition | 0.32 | % | ALA4887778 | Not Active | % | Homo sapiens | |||
8. | ALA4580220 | EUB0000311 | % residual kinase activity | 99 | % | ALA4884528 | Not Active | % | Homo sapiens | |||
9. | BAY-885 | BAY-885; 41 | % residual kinase activity | 107 | % | ALA4881290 | Not Active | % | Homo sapiens | |||
10. | KU 60019 | SID124939250 | IC50 | = | 6 | nM | ALA3395883 | 8.22 | nM | Homo sapiens | ||
11. | ALA3315358 | 9a, YQL-9a | Activity | 0 | ALA3371179 | Active | Homo sapiens | |||||
12. | ALA3315358 | 9a, YQL-9a | Activity | 0 | ALA3371178 | Active | Homo sapiens | |||||
13. | ALA3315358 | 9a, YQL-9a | Activity | 0 | ALA3371177 | Active | Homo sapiens | |||||
14. | ALA3315358 | 9a, YQL-9a | Activity | 0 | ALA3371176 | Active | Homo sapiens | |||||
15. | ETP-46464 | 15, ETP-46464 | IC50 | > | 36 | nM | ALA3374531 | nM | Homo sapiens | |||
16. | ALA3355480 | 13 | IC50 | = | 15 | uM | ALA3372426 | 4.82 | nM | Homo sapiens | ||
17. | ALA3355474 | 7 | INH | 0 | ALA3372409 | Not Active | % | Homo sapiens | ||||
18. | ALA3355074 | 7 | IC50 | = | 4.3 | uM | ALA3379629 | 5.37 | nM | Homo sapiens | ||
19. | ALA3355073 | 6 | IC50 | = | 14 | uM | ALA3379629 | 4.85 | nM | Homo sapiens | ||
20. | ALA3355072 | 5 | IC50 | = | 0.13 | uM | ALA3379629 | 6.89 | nM | Homo sapiens |