# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA241253 | 21g | IC50 | = | 40 | nmol/L | ALA2149804 | 7.40 | nM | Homo sapiens | ||
2. | ALA391466 | 17g | IC50 | = | 12 | nmol/L | ALA2149804 | 7.92 | nM | Homo sapiens | ||
3. | ALA2147771 | 8p | IC50 | = | 220 | nmol/L | ALA2149804 | 6.66 | nM | Homo sapiens | ||
4. | ALA2147712 | 8j | IC50 | = | 86 | nmol/L | ALA2149804 | 7.07 | nM | Homo sapiens | ||
5. | Teneligliptin | 8g, teneligliptin | IC50 | = | 260 | nmol/L | ALA2149804 | 6.58 | nM | Homo sapiens | ||
6. | sitagliptin | Sitagliptin | IC50 | = | 48000 | nM | ALA2149438 | 4.32 | nM | Homo sapiens | ||
7. | Alogliptin | 10, alogliptin, SYR-322 | IC50 | > | 100000 | nM | ALA2149438 | nM | Homo sapiens | |||
8. | Linagliptin | 1, BI 1356 | IC50 | > | 40000 | nM | ALA2149438 | nM | Homo sapiens | |||
9. | Saxagliptin | 26 | IC50 | = | 244 | nM | ALA2149438 | 6.61 | nM | Homo sapiens | ||
10. | Vildagliptin (LAF-237) | 2 | Ki | = | 810 | nM | ALA2149438 | 6.09 | nM | Homo sapiens | ||
11. | ALA2147070 | 28 | IC50 | > | 100000 | nM | ALA2149438 | nM | Homo sapiens | |||
12. | ALA3127991 | 6m | IC50 | = | 0.7 | uM | ALA3128755 | 6.16 | nM | Homo sapiens | ||
13. | ALA3127988 | 6j | IC50 | = | 0.9 | uM | ALA3128755 | 6.05 | nM | Homo sapiens | ||
14. | ALA3127989 | 6k | IC50 | = | 1 | uM | ALA3128755 | 6.00 | nM | Homo sapiens | ||
15. | ALA3127990 | 6l | IC50 | = | 1.3 | uM | ALA3128755 | 5.89 | nM | Homo sapiens | ||
16. | ALA3127984 | 6f | IC50 | = | 1.4 | uM | ALA3128755 | 5.85 | nM | Homo sapiens | ||
17. | ALA3127986 | 6h | IC50 | = | 1.8 | uM | ALA3128755 | 5.75 | nM | Homo sapiens | ||
18. | ALA3127987 | 6i | IC50 | = | 3.3 | uM | ALA3128755 | 5.48 | nM | Homo sapiens | ||
19. | ALA3127985 | 6g | IC50 | = | 3.4 | uM | ALA3128755 | 5.47 | nM | Homo sapiens | ||
20. | ALA3127992 | 6n | IC50 | = | 4.7 | uM | ALA3128755 | 5.33 | nM | Homo sapiens |