# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2441828 | 1a | Ki | = | 3.4 | nM | ALA2444438 | 8.47 | nM | Homo sapiens | ||
2. | ALA2441829 | 1b | Ki | = | 1.3 | nM | ALA2444438 | 8.89 | nM | Homo sapiens | ||
3. | ALA2441830 | 1c | Ki | = | 5.4 | nM | ALA2444438 | 8.27 | nM | Homo sapiens | ||
4. | ALA2441830 | 1c | Ki | = | 2.3 | nM | ALA2444438 | 8.64 | nM | Homo sapiens | ||
5. | ALA2441830 | 1c | Ki | > | 30 | nM | ALA2444438 | nM | Homo sapiens | |||
6. | ALA2441831 | 2b, more active atropisomer | Ki | = | 1.2 | nM | ALA2444438 | 8.92 | nM | Homo sapiens | ||
7. | ALA2441832 | 1d | Ki | > | 10 | nM | ALA2444438 | nM | Homo sapiens | |||
8. | ALA2441833 | 2c, More active atropisomer | Ki | = | 3.7 | nM | ALA2444438 | 8.43 | nM | Homo sapiens | ||
9. | ALA2441834 | 2d, More active atropisomer | Ki | = | 7.3 | nM | ALA2444438 | 8.14 | nM | Homo sapiens | ||
10. | ALA2441835 | 2e, More active atropisomer | Ki | = | 4.3 | nM | ALA2444438 | 8.37 | nM | Homo sapiens | ||
11. | ALA2441836 | 1e, BMS-744891 | Ki | = | 4.6 | nM | ALA2444438 | 8.34 | nM | Homo sapiens | ||
12. | ALA2441836 | 1e, BMS-744891 | Ki | = | 1.9 | nM | ALA2444438 | 8.72 | nM | Homo sapiens | ||
13. | ALA2441836 | 1e, BMS-744891 | Ki | > | 30 | nM | ALA2444438 | nM | Homo sapiens | |||
14. | ALA2441837 | 2g, More active atropisomer | Ki | = | 2.3 | nM | ALA2444438 | 8.64 | nM | Homo sapiens | ||
15. | ALA2441837 | 2g, More active atropisomer | Ki | > | 30 | nM | ALA2444438 | nM | Homo sapiens | |||
16. | ALA2441838 | 2h, More active atropisomer | Ki | = | 3.1 | nM | ALA2444438 | 8.51 | nM | Homo sapiens | ||
17. | ALA2441839 | 2i, More active atropisomer | Ki | = | 0.5 | nM | ALA2444438 | 9.30 | nM | Homo sapiens | ||
18. | ALA2441840 | 2j, More active atropisomer | Ki | > | 30 | nM | ALA2444438 | nM | Homo sapiens | |||
19. | ALA2441841 | 2k, More active atropisomer | Ki | = | 2.9 | nM | ALA2444438 | 8.54 | nM | Homo sapiens | ||
20. | ALA2441842 | 1f | Ki | > | 30 | nM | ALA2444438 | nM | Homo sapiens |