# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | CEP-1347 | 2 | INH | > | 99 | % | ALA2438993 | % | Homo sapiens | |||
2. | URMC-099 | 1, URMC-099 | IC50 | = | 290 | nM | ALA2439769 | 6.54 | nM | Homo sapiens | ||
3. | ALA2425654 | 3 | INH | < | 50 | % | ALA2428025 | % | Homo sapiens | |||
4. | ALA2425652 | 4 | INH | = | 97 | % | ALA2428025 | % | Homo sapiens | |||
5. | ALA2425649 | 8 | INH | < | 50 | % | ALA2428025 | % | Homo sapiens | |||
6. | ALA2425645 | 11 | INH | < | 50 | % | ALA2428025 | % | Homo sapiens | |||
7. | ALA2425644 | 13 | INH | = | 96 | % | ALA2428025 | % | Homo sapiens | |||
8. | ALA2425646 | 12 | INH | < | 50 | % | ALA2428025 | % | Homo sapiens | |||
9. | ALA2420899 | 41 | INH | = | 54 | % | ALA2423808 | % | Homo sapiens | |||
10. | ALA2420900 | 42 | INH | = | 46 | % | ALA2423808 | % | Homo sapiens | |||
11. | ALA2420901 | 45 | INH | = | 61 | % | ALA2423808 | % | Homo sapiens | |||
12. | ALA2402081 | 37 | INH | = | 1 | % | ALA2405952 | % | Homo sapiens | |||
13. | ALA2398657 | 27, IBPR001 | INH | > | 50 | % | ALA2400109 | % | Homo sapiens | |||
14. | Tozasertib | VX-680 | Ki | = | 4.6 | nM | ALA2396195 | 8.34 | nM | Homo sapiens | ||
15. | ALA2386796 | 9p | INH | = | 16 | % | ALA2389848 | % | Homo sapiens | |||
16. | ALA2386802 | 10f | INH | 0 | ALA2389848 | Not Determined | % | Homo sapiens | ||||
17. | ALA2380586 | 32a | INH | > | 50 | % | ALA2383378 | % | Homo sapiens | |||
18. | ALA2380587 | 32b | INH | > | 50 | % | ALA2383378 | % | Homo sapiens | |||
19. | ZM-447439 | 2 | INH | > | 50 | % | ALA2091235 | % | Homo sapiens | |||
20. | TPCA-1 | Calbio IV | INH | > | 25 | % | ALA2091235 | % | Homo sapiens |