# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4639128 | 62 | pIC50 | < | 4.3 | ALA5303907 | nM | Homo sapiens | ||||
2. | GSK620 | 1; 20 | pIC50 | < | 4.3 | ALA5303858 | nM | Homo sapiens | ||||
3. | GSK046 | 15; GSK046 | pIC50 | < | 4.3 | ALA5303809 | nM | Homo sapiens | ||||
4. | ALA219631 | CI-1041 | Ki | = | 30 | nM | ALA3804511 | 7.52 | nM | Homo sapiens | ||
5. | ALA3798280 | 28 | INH | = | 0 | % | ALA3804513 | % | Homo sapiens | |||
6. | ALA3798610 | trans-27 | INH | = | 18 | % | ALA3804513 | % | Homo sapiens | |||
7. | ALA3797211 | cis-26 | INH | = | 0 | % | ALA3804513 | % | Homo sapiens | |||
8. | Eliprodil | (rac)-9 | Ki | = | 13 | nM | ALA3804512 | 7.89 | nM | Homo sapiens | ||
9. | ALA319706 | 19 | Ki | = | 10 | nM | ALA3804512 | 8.00 | nM | Homo sapiens | ||
10. | ALA3797704 | 30 | Ki | = | 697 | nM | ALA3804512 | 6.16 | nM | Homo sapiens | ||
11. | I-BRD9 | 45; I-BRD9 | INH | 0 | ALA3773852 | Not Active | % | Homo sapiens | ||||
12. | ALA3357784 | 5 | Ki | = | 10 | nM | ALA3737377 | 8.00 | nM | Homo sapiens | ||
13. | Eliprodil | (rac)-9 | Ki | = | 13 | nM | ALA3737377 | 7.89 | nM | Homo sapiens | ||
14. | ALA319706 | 19 | Ki | = | 10 | nM | ALA3737377 | 8.00 | nM | Homo sapiens | ||
15. | ALA3736502 | 8d | Ki | = | 3.8 | nM | ALA3737377 | 8.42 | nM | Homo sapiens | ||
16. | ALA3735947 | 8c | Ki | = | 1.6 | nM | ALA3737377 | 8.80 | nM | Homo sapiens | ||
17. | ALA3735485 | 8b | Ki | = | 3.3 | nM | ALA3737377 | 8.48 | nM | Homo sapiens | ||
18. | ALA3735173 | 8a | Ki | = | 7.6 | nM | ALA3737377 | 8.12 | nM | Homo sapiens | ||
19. | EVT-101 free base | EVT-101 | IC50 | = | 17 | nM | ALA5255361 | 7.77 | nM | Homo sapiens | ||
20. | CP-101,606 | 1 | IC50 | = | 11 | nM | ALA5255361 | 7.96 | nM | Homo sapiens |