# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5278465 | 33 | IC50 | > | 50 | uM | ALA5252890 | nM | Homo sapiens | |||
2. | ALA5288565 | 29 | IC50 | > | 50 | uM | ALA5252890 | nM | Homo sapiens | |||
3. | ALA5270581 | 18 | IC50 | > | 50 | uM | ALA5252890 | nM | Homo sapiens | |||
4. | ALA4213175 | Fig S3, Cpd 6 | IC50 | > | 50 | uM | ALA5252890 | nM | Homo sapiens | |||
5. | BAW2881(NVP-BAW2881) | 2 | IC50 | = | 30 | nM | ALA5252779 | 7.52 | nM | Homo sapiens | ||
6. | BFH772 | 1 | IC50 | = | 30 | nM | ALA5252779 | 7.52 | nM | Homo sapiens | ||
7. | BFH772 | 1 | IC50 | > | 2 | uM | ALA5252752 | nM | Homo sapiens | |||
8. | BAW2881(NVP-BAW2881) | 2 | IC50 | > | 10 | uM | ALA5252752 | nM | Homo sapiens | |||
9. | ALA5270781 | 38 | IC50 | > | 50 | uM | ALA5252065 | nM | Homo sapiens | |||
10. | ALA5267815 | 12a | INH | 0 | ALA5244017 | Not Active | % | Homo sapiens | ||||
11. | Ripretinib (DCC-2618) | 4; DCC-2618 | IC50 | = | 25 | uM | ALA5238316 | 4.60 | nM | Homo sapiens | ||
12. | Ripretinib (DCC-2618) | 4; DCC-2618 | IC50 | = | 9.2 | nM | ALA5238315 | 8.04 | nM | Homo sapiens | ||
13. | Pexidartinib | PEXIDARTINIB | IC50 | = | 27 | nM | ALA5238314 | 7.57 | nM | Homo sapiens | ||
14. | AZD3229 | 44; AZD3229 | IC50 | = | 3 | nM | ALA5238314 | 8.52 | nM | Homo sapiens | ||
15. | Ripretinib (DCC-2618) | 4; DCC-2618 | IC50 | = | 13 | nM | ALA5238314 | 7.89 | nM | Homo sapiens | ||
16. | Imatinib (STI571) | 1 | IC50 | = | 400 | nM | ALA5233738 | 6.40 | nM | Homo sapiens | ||
17. | ALA5267404 | 12 | IC50 | = | 7471 | nM | ALA5225629 | 5.13 | nM | Homo sapiens | ||
18. | ALA5289612 | 11 | IC50 | = | 1976 | nM | ALA5225629 | 5.70 | nM | Homo sapiens | ||
19. | ALA5275738 | 10 | IC50 | = | 1078 | nM | ALA5225629 | 5.97 | nM | Homo sapiens | ||
20. | ALA5281791 | 9 | IC50 | = | 857 | nM | ALA5225629 | 6.07 | nM | Homo sapiens |