# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Bestatin | bestatin | IC50 | = | 2.5 | uM | ALA2415687 | 5.60 | nM | Homo sapiens | ||
2. | ALA116438 | 15 | IC50 | = | 10 | uM | ALA2415687 | 5.00 | nM | Homo sapiens | ||
3. | ALA2393088 | 2, LB-4b | IC50 | = | 3 | uM | ALA2395150 | 5.52 | nM | Homo sapiens | ||
4. | Bestatin | bestatin | IC50 | = | 40 | uM | ALA2395150 | 4.40 | nM | Homo sapiens | ||
5. | ALA2393088 | 2, LB-4b | Ratio IC50 | = | 10 | ALA2394983 | Homo sapiens | |||||
6. | ALA1941150 | Probestin | Ki | = | 19 | nM | ALA2395658 | 7.72 | nM | Homo sapiens | ||
7. | ALA2376104 | 10a | IC50 | = | 9.58 | uM | ALA2379683 | 5.02 | nM | Homo sapiens | ||
8. | ALA2376105 | 10b | IC50 | = | 16.19 | uM | ALA2379683 | 4.79 | nM | Homo sapiens | ||
9. | ALA1712297 | SID47195051 | IC50 | = | 12.4 | uM | ALA2379683 | 4.91 | nM | Homo sapiens | ||
10. | ALA2376108 | 11a | IC50 | = | 10.94 | uM | ALA2379683 | 4.96 | nM | Homo sapiens | ||
11. | ALA2376109 | 11b | IC50 | = | 97.49 | uM | ALA2379683 | 4.01 | nM | Homo sapiens | ||
12. | ALA2376110 | 11c | IC50 | = | 19.66 | uM | ALA2379683 | 4.71 | nM | Homo sapiens | ||
13. | ALA2376113 | 12a | IC50 | = | 3.12 | uM | ALA2379683 | 5.51 | nM | Homo sapiens | ||
14. | ALA2376114 | 12b | IC50 | = | 15.16 | uM | ALA2379683 | 4.82 | nM | Homo sapiens | ||
15. | ALA2376115 | 12c | IC50 | = | 12.1 | uM | ALA2379683 | 4.92 | nM | Homo sapiens | ||
16. | Bestatin | bestatin | IC50 | = | 29.67 | uM | ALA2379683 | 4.53 | nM | Homo sapiens | ||
17. | ALA1668626 | 4 | Ki | = | 2 | uM | ALA2353230 | 5.70 | nM | Homo sapiens | ||
18. | ALA1821978 | 1f | Ki | = | 11 | nM | ALA2353230 | 7.96 | nM | Homo sapiens | ||
19. | 7-amino-1-bromo-4-phenyl-5,7,8,9-tetrahydrobenzo[7]annulen-6-one | I3 | Ki | = | 0.35 | nM | ALA2353230 | 9.46 | nM | Homo sapiens | ||
20. | 7-amino-1-bromo-4-phenyl-5,7,8,9-tetrahydrobenzo[7]annulen-6-one | I3 | INH | 0 | ALA2352975 | Active | % | Homo sapiens |