# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | VU 0409106 | 24, VU0409106 | INH | > | 35 | % | ALA2446046 | % | Homo sapiens | |||
2. | ML315 | SID124360160 | INH | = | 3 | % | ALA2396437 | % | Homo sapiens | |||
3. | ALA437472 | ET-1 | IC50 | = | 5 | 10'-11M | ALA2395695 | 10.30 | nM | Homo sapiens | ||
4. | ALA437472 | ET-1 | Ki | = | 2.5 | 10'-11M | ALA2395695 | 10.60 | nM | Homo sapiens | ||
5. | ALA437472 | ET-1 | INH | = | 3 | % | ALA2396217 | % | Homo sapiens | |||
6. | ALA437472 | ET-1 | IC50 | = | 0.23 | nM | ALA2395270 | 9.64 | nM | Homo sapiens | ||
7. | ALA437472 | ET-1 | Ki | = | 0.14 | nM | ALA2395270 | 9.85 | nM | Homo sapiens | ||
8. | E1R | E1R, 4R,5S-2a | INH | = | -2 | % | ALA2393948 | % | Homo sapiens | |||
9. | ALA437472 | ET-1 | IC50 | = | 0.11 | nM | ALA2395015 | 9.96 | nM | Homo sapiens | ||
10. | ALA2392692 | 27, GSK2188931B | INH | < | 50 | % | ALA2395859 | % | Homo sapiens | |||
11. | ALA2326501 | 5d | INH | = | 14 | % | ALA2329406 | % | Homo sapiens | |||
12. | ALA2296888 | 1 | IC50 | = | 11 | uM | ALA3075855 | 4.96 | nM | Homo sapiens | ||
13. | ALA2296889 | 2 | IC50 | = | 3.8 | uM | ALA3075855 | 5.42 | nM | Homo sapiens | ||
14. | BQ-123 | BQ-123 | IC50 | = | 37 | nM | ALA3074523 | 7.43 | nM | Homo sapiens | ||
15. | ALA2261359 | 7a | Kb | = | 2 | nM | ALA3057240 | nM | Homo sapiens | |||
16. | ALA22513 | 32 | IC50 | = | 0.55 | nM | ALA3056377 | 9.26 | nM | Homo sapiens | ||
17. | ALA23833 | 18 | IC50 | = | 32 | nM | ALA3056377 | 7.50 | nM | Homo sapiens | ||
18. | ALA262784 | 9 | IC50 | = | 2.3 | nM | ALA3056377 | 8.64 | nM | Homo sapiens | ||
19. | ALA2261356 | 4 | IC50 | = | 560 | nM | ALA3056377 | 6.25 | nM | Homo sapiens | ||
20. | ALA2261357 | 5 | IC50 | = | 1.7 | nM | ALA3056377 | 8.77 | nM | Homo sapiens |