| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5078078 | T-036 | IC50 | > | 10 | uM | ALA5304946 | nM | Homo sapiens | |||
| 2. | ALA5078078 | T-036 | EC50 | > | 10 | uM | ALA5304945 | nM | Homo sapiens | |||
| 3. |  ALA5306577 | EUB0002354 | Inhibition | = | 3 | % | ALA5304423 | % | Homo sapiens | |||
| 4. |  ALA5303444 | EUB0001742a | % Ctrl | = | 111 | % | ALA5304335 | Not Active | % | Homo sapiens | ||
| 5. |  BI-3812 | 44 | % Ctrl | = | 104 | % | ALA5304237 | Not Active | % | Homo sapiens | ||
| 6. |  BI-3802 | BI-3802 | % Ctrl | = | 100 | % | ALA5304133 | Not Active | % | Homo sapiens | ||
| 7. |  ALA5306038 | EUB0001699 | % Ctrl | = | 104 | % | ALA5304087 | Not Active | % | Homo sapiens | ||
| 8. |  ALA5303508 | EUB0001755aCl | % Ctrl | = | 100 | % | ALA5304041 | Not Active | % | Homo sapiens | ||
| 9. |  ALA5308145 | EUB0002187 | % Ctrl | = | 104 | % | ALA5303991 | Not Active | % | Homo sapiens | ||
| 10. |  ALA5307400 | EUB0002188 | % Ctrl | = | 97 | % | ALA5303947 | Not Active | % | Homo sapiens | ||
| 11. |  ALA4533479 | EUB0000339 | IC50 | = | 1.6 | uM | ALA5058654 | 5.80 | Not Active | nM | Homo sapiens | |
| 12. |  ALA3775769 | 23a | INH | = | -4.4 | % | ALA3778199 | % | Homo sapiens | |||
| 13. |  ALA3775436 | 22a | INH | = | -3.4 | % | ALA3778199 | % | Homo sapiens | |||
| 14. |  endothelin-1 | Endothelin-1 | IC50 | = | 2.3 | 10'-11M | ALA3779717 | 10.64 | nM | Homo sapiens | ||
| 15. |  (S)-ARN2508 | (+)-10r | Activity | = | -6.2 | % | ALA3779477 | % | Homo sapiens | |||
| 16. |  ALA3771118 | 4a; PF-06761281 | INH | 0 | ALA3773639 | Not Active | % | Homo sapiens | ||||
| 17. |  ALA3763166 | 40 | INH | < | 50 | % | ALA3766819 | % | Homo sapiens | |||
| 18. |  Bosentan | Bosentan | IC50 | = | 8.4 | nM | ALA3757818 | 8.08 | nM | Homo sapiens | ||
| 19. |  ALA3753047 | 1w | IC50 | > | 20000 | nM | ALA3757818 | nM | Homo sapiens | |||
| 20. |  ALA3753277 | 1v | IC50 | = | 11000 | nM | ALA3757818 | 4.96 | nM | Homo sapiens |
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