# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2442940 | 10d | INH | 0 | ALA2446834 | Not Active | % | Homo sapiens | ||||
2. | VU 0409106 | 24, VU0409106 | INH | > | 35 | % | ALA2446040 | % | Homo sapiens | |||
3. | ALA384467 | 9 | EC50 | = | 1.1 | nM | ALA2428211 | 8.96 | nM | Homo sapiens | ||
4. | ALA384467 | 9 | Ki | = | 1.2 | nM | ALA2428212 | 8.92 | nM | Homo sapiens | ||
5. | ALA1801004 | 22 | Ki | = | 1.1 | nM | ALA2428212 | 8.96 | nM | Homo sapiens | ||
6. | ALA2426658 | (3S)-5a | Ki | = | 2.7 | nM | ALA2428212 | 8.57 | nM | Homo sapiens | ||
7. | ALA2426659 | (3R)-5a | Ki | = | 13 | nM | ALA2428212 | 7.89 | nM | Homo sapiens | ||
8. | ALA2426660 | 5b | Ki | = | 5 | nM | ALA2428212 | 8.30 | nM | Homo sapiens | ||
9. | ALA2426661 | 5c | Ki | = | 18 | nM | ALA2428212 | 7.75 | nM | Homo sapiens | ||
10. | ALA2426662 | (3S)-5c | Ki | = | 5.1 | nM | ALA2428212 | 8.29 | nM | Homo sapiens | ||
11. | ALA2426663 | (3R)-5c | Ki | = | 6.7 | nM | ALA2428212 | 8.17 | nM | Homo sapiens | ||
12. | ALA2426664 | 5d | Ki | = | 15 | nM | ALA2428212 | 7.82 | nM | Homo sapiens | ||
13. | ALA2426665 | (3S)-5d | Ki | = | 6 | nM | ALA2428212 | 8.22 | nM | Homo sapiens | ||
14. | ALA2426644 | (3R)-5d | Ki | = | 7.9 | nM | ALA2428212 | 8.10 | nM | Homo sapiens | ||
15. | ALA2426645 | 5e | Ki | = | 18 | nM | ALA2428212 | 7.75 | nM | Homo sapiens | ||
16. | ALA2426646 | 5f | Ki | = | 29 | nM | ALA2428212 | 7.54 | nM | Homo sapiens | ||
17. | ALA2426647 | 5g | Ki | = | 8.1 | nM | ALA2428212 | 8.09 | nM | Homo sapiens | ||
18. | ALA2426648 | (3S)-5h | Ki | = | 0.9 | nM | ALA2428212 | 9.05 | nM | Homo sapiens | ||
19. | ALA2426649 | (3R)-5h | Ki | = | 4 | nM | ALA2428212 | 8.40 | nM | Homo sapiens | ||
20. | ALA2426650 | 5i | Ki | = | 1.9 | nM | ALA2428212 | 8.72 | nM | Homo sapiens |