# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5306577 | EUB0002354 | Inhibition | = | -7 | % | ALA5304477 | % | Homo sapiens | |||
2. | ALA4639128 | 62 | pIC50 | < | 4.6 | ALA5303905 | nM | Homo sapiens | ||||
3. | GSK620 | 1; 20 | pIC50 | < | 4.6 | ALA5303856 | nM | Homo sapiens | ||||
4. | GSK046 | 15; GSK046 | pIC50 | < | 4.6 | ALA5303808 | nM | Homo sapiens | ||||
5. | AM 0902 | 27; AM-0902 | Activity | > | 77 | % | ALA3789369 | % | Homo sapiens | |||
6. | ALA3780686 | 14 | Ki | = | 6.72 | nM | ALA3783010 | 8.17 | nM | Homo sapiens | ||
7. | ALA3781336 | 13 | Ki | = | 7.54 | nM | ALA3783010 | 8.12 | nM | Homo sapiens | ||
8. | ALA3781519 | 12 | Ki | = | 8.11 | nM | ALA3783010 | 8.09 | nM | Homo sapiens | ||
9. | ALA3780818 | 11 | Ki | = | 8.33 | nM | ALA3783010 | 8.08 | nM | Homo sapiens | ||
10. | ALA3781680 | 10 | Ki | 0 | ALA3783010 | Not Determined | Homo sapiens | |||||
11. | ALA3780408 | 9 | Ki | 0 | ALA3783010 | Not Determined | Homo sapiens | |||||
12. | ALA3780820 | 8 | Ki | 0 | ALA3783010 | Not Determined | Homo sapiens | |||||
13. | ALA3780776 | 7 | Ki | 0 | ALA3783010 | Not Determined | Homo sapiens | |||||
14. | ALA3408519 | 22, H-Dmt-D-Arg-Aba-beta-Ala-NMe-Bn | Ki | = | 6.44 | nM | ALA3783010 | 8.19 | nM | Homo sapiens | ||
15. | ALA1782141 | 35 | Ki | = | 7.8 | nM | ALA3783010 | 8.11 | nM | Homo sapiens | ||
16. | ALA3780686 | 14 | Ki | = | 1.9 | nM | ALA3782901 | 8.72 | nM | Homo sapiens | ||
17. | ALA3781336 | 13 | Ki | = | 1.4 | nM | ALA3782901 | 8.85 | nM | Homo sapiens | ||
18. | ALA3781519 | 12 | Ki | = | 1.4 | nM | ALA3782901 | 8.85 | nM | Homo sapiens | ||
19. | ALA3780818 | 11 | Ki | = | 2.2 | nM | ALA3782901 | 8.66 | nM | Homo sapiens | ||
20. | ALA3781680 | 10 | Ki | 0 | ALA3782901 | Not Determined | Homo sapiens |