# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5273129 | (5S,6R,9S)-316 | Activity | = | 47 | % | ALA5247083 | % | Homo sapiens | |||
2. | ALA5268226 | (5S,6S,9R)-316 | Activity | = | 44 | % | ALA5247083 | % | Homo sapiens | |||
3. | ALA5283681 | (5S,6R,9R)-316 | IC50 | = | 400 | nM | ALA5247052 | 6.40 | nM | Homo sapiens | ||
4. | ALA5290533 | 320 | IC50 | = | 0.1 | nM | ALA5247052 | 10.00 | nM | Homo sapiens | ||
5. | ALA5286807 | 319 | IC50 | = | 24 | nM | ALA5247052 | 7.62 | nM | Homo sapiens | ||
6. | ALA5285318 | 318 | IC50 | = | 1.4 | nM | ALA5247052 | 8.85 | nM | Homo sapiens | ||
7. | ALA5284869 | 317 | IC50 | = | 1.1 | nM | ALA5247052 | 8.96 | nM | Homo sapiens | ||
8. | ALA5291459 | 316 | IC50 | = | 28 | nM | ALA5247052 | 7.55 | nM | Homo sapiens | ||
9. | Aprepitant | 2 | IC50 | = | 0.09 | nM | ALA5247052 | 10.05 | nM | Homo sapiens | ||
10. | ALA52330 | 1 | IC50 | = | 0.09 | nM | ALA5247052 | 10.05 | nM | Homo sapiens | ||
11. | ALA99055 | 12 | IC50 | = | 0.05 | nM | ALA5247052 | 10.30 | nM | Homo sapiens | ||
12. | ALA27006 | 2 | IC50 | = | 0.87 | nM | ALA5247052 | 9.06 | nM | Homo sapiens | ||
13. | ALA140745 | 16 | IC50 | = | 0.07 | nM | ALA5244908 | 10.15 | nM | Homo sapiens | ||
14. | Aprepitant | 2 | IC50 | = | 0.09 | nM | ALA5244908 | 10.05 | nM | Homo sapiens | ||
15. | PF 05105679 | 8, PF-05105679 | % of effect | = | 18 | % | ALA5214516 | % | Homo sapiens | |||
16. | ALA3736287 | 12 | Ki | = | 2.2 | nM | ALA5145925 | 8.66 | nM | Homo sapiens | ||
17. | GSK-2894631A | 1bv | INH | 0 | ALA4402267 | Not Active | % | Homo sapiens | ||||
18. | Pemigatinib | PEMIGATINIB | INH | 0 | ALA4810248 | Not Active | % | Homo sapiens | ||||
19. | ALA4794099 | stearyl-CMSP | Activity | 0 | ALA4726518 | Active | Homo sapiens | |||||
20. | ALA4750714 | stearyl-CAMEL | Activity | 0 | ALA4726518 | Not Active | Homo sapiens |