# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5306577 | EUB0002354 | Inhibition | = | -15 | % | ALA5304469 | % | Homo sapiens | |||
2. | ALA3765778 | 27 | Ki | = | 2 | uM | ALA3769214 | 5.70 | nM | Homo sapiens | ||
3. | ALA3746457 | 4k | INH | = | 57 | % | ALA3749991 | % | Homo sapiens | |||
4. | ALA3186763 | SID144087340 | INH | = | 7.04 | % | ALA3383691 | % | Homo sapiens | |||
5. | SX-517 | 7, SX-517 | IC50 | > | 5000 | nM | ALA3387790 | nM | Homo sapiens | |||
6. | ALA3958704 | 8a | INH | < | 20 | % | ALA4184489 | % | Homo sapiens | |||
7. | Morphothiadin | 5; GLS4 | INH | = | 10 | % | ALA4177953 | % | Homo sapiens | |||
8. | VU 6005649 | 9f; VU6005649 | INH | < | 50 | % | ALA4140876 | % | Homo sapiens | |||
9. | ALA4172540 | 19; VU6010572, (S)-enantiomer | INH | > | 50 | % | ALA4134117 | % | Homo sapiens | |||
10. | ALA4089114 | 51 | INH | = | 55 | % | ALA4047844 | % | Homo sapiens | |||
11. | ALA4086541 | (S)-28b | INH | 0 | ALA4044978 | Not Active | % | Homo sapiens | ||||
12. | ALA3288123 | 15 | Activity | 0 | ALA3291825 | Not Active | Homo sapiens | |||||
13. | AZD 1283 | 3, AZD1283 | Activity | 0 | ALA3291825 | Not Active | Homo sapiens | |||||
14. | ALA4793451 | 4j; MGS0274 | Activity | 0 | ALA4708816 | Not Active | Homo sapiens | |||||
15. | ALA334014 | 3 | Activity | 0 | ALA4708816 | Not Active | Homo sapiens | |||||
16. | ALA4754102 | 8; VU6014181 | INH | < | 50 | % | ALA4671124 | % | Homo sapiens | |||
17. | ALA4761695 | 21a; VU06027459 | INH | < | 50 | % | ALA4671124 | % | Homo sapiens | |||
18. | ALA4795177 | 21g; VU6005806; AZN-00016130 | Activity | > | 50 | % | ALA4667540 | % | Homo sapiens | |||
19. | ALA4097778 | 16h | % inhibition | -24 | % | ALA4884611 | Not Active | % | Homo sapiens | |||
20. | ALA4549667 | EUB0000720 | % inhibition | -27 | % | ALA4884611 | Not Active | % | Homo sapiens |