# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5280210 | 31 | INH | = | 64 | % | ALA5236910 | % | Homo sapiens | |||
2. | ALA2112095 | 5d | Ki | > | 100000 | nM | ALA5233317 | nM | Homo sapiens | |||
3. | ALA5274986 | (N)-mc Ado | Ki | = | 22500 | nM | ALA5233317 | 4.65 | nM | Homo sapiens | ||
4. | Caffeine | caffeine | pKi | = | 4.3 | ALA5223689 | 4.30 | nM | Homo sapiens | |||
5. | Caffeine | caffeine | IC50 | = | 9.6 | uM | ALA5223689 | 5.02 | nM | Homo sapiens | ||
6. | Theobromine | theobromine | IC50 | > | 250 | uM | ALA5223689 | nM | Homo sapiens | |||
7. | Theobromine | theobromine | Ki | > | 250 | uM | ALA5223684 | nM | Homo sapiens | |||
8. | WM 1119 | 4; WM-1119 | % of inhibition | = | 49 | % | ALA5214066 | % | Homo sapiens | |||
9. | A 196 | A-196 | Ki | = | 28 | nM | ALA5214592 | 7.55 | nM | Homo sapiens | ||
10. | A 196 | A-196 | % of inhibition | = | 98 | % | ALA5214591 | % | Homo sapiens | |||
11. | BIX 02565 | 24, BIX 02565, eutamer | IC50 | = | 1420 | nM | ALA5213133 | 5.85 | nM | Homo sapiens | ||
12. | ALA5200705 | 26 | Activity | = | -31.2 | % | ALA5164143 | % | Homo sapiens | |||
13. | ALA5200705 | 26 | Activity | = | -0.3 | % | ALA5164119 | % | Homo sapiens | |||
14. | ALA5204735 | 36b | Ki | = | 74.3 | nM | ALA5163974 | 7.13 | nM | Homo sapiens | ||
15. | ALA5195323 | 36a | Ki | = | 15 | nM | ALA5163974 | 7.82 | nM | Homo sapiens | ||
16. | ALA5171672 | 30l | Ki | = | 159.3 | nM | ALA5163974 | 6.80 | nM | Homo sapiens | ||
17. | ALA5189321 | 30k | Ki | = | 72.8 | nM | ALA5163974 | 7.14 | nM | Homo sapiens | ||
18. | ALA5179716 | 30j | Ki | = | 72 | nM | ALA5163974 | 7.14 | nM | Homo sapiens | ||
19. | ALA5188801 | 30i | Ki | = | 14.7 | nM | ALA5163974 | 7.83 | nM | Homo sapiens | ||
20. | ALA5188108 | 30h | Ki | = | 68.3 | nM | ALA5163974 | 7.17 | nM | Homo sapiens |