# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2385460 | 26, AM-5262 | INH | < | 70 | % | ALA2388540 | % | Homo sapiens | |||
2. | ALA2385464 | 30 | INH | < | 70 | % | ALA2388540 | % | Homo sapiens | |||
3. | AM-1638 | 21, AM-1638 | INH | > | 70 | % | ALA2388540 | % | Homo sapiens | |||
4. | PQCA | 4i | % inhibition | 13 | % | ALA4882985 | Not Active | % | Homo sapiens | |||
5. | THPP-1 | THPP-1 | % inhibition | 7 | % | ALA4882985 | Not Active | % | Homo sapiens | |||
6. | PPTN | 2 | % inhibition | -19 | % | ALA4882985 | Not Active | % | Homo sapiens | |||
7. | MLI-2 | 1; MLi-2 | % inhibition | -14 | % | ALA4882985 | Not Active | % | Homo sapiens | |||
8. | Remibrutinib (LOU064) | 25; LOU064 | Activity | 0 | ALA4358665 | Not Active | Homo sapiens | |||||
9. | CHDI 00390576 | 22 | INH | < | 25 | % | ALA4311080 | % | Homo sapiens | |||
10. | ALA4437833 | 16 | INH | < | 25 | % | ALA4311080 | % | Homo sapiens | |||
11. | (S)-ARN2508 | (+)-10r | Activity | = | -14.9 | % | ALA3777183 | % | Homo sapiens | |||
12. | ALA5090753 | RgIA-5524 | Activity | = | -4 | % | ALA5034717 | % | Homo sapiens | |||
13. | ALA2206397 | 6d, Ro-4992479 | INH | = | 0 | % | ALA2213034 | % | Homo sapiens | |||
14. | ALA1717527 | SID49724559 | Potency | 2.909 | uM | ALA1737857 | inconclusive | nM | Homo sapiens | |||
15. | ALA1727220 | SID49671070 | Potency | 0.018 | uM | ALA1737857 | inconclusive | nM | Homo sapiens | |||
16. | ALA1447664 | SID24832136 | Potency | 0.013 | uM | ALA1737857 | inconclusive | nM | Homo sapiens | |||
17. | ALA1472277 | SID49680356 | Potency | 0.023 | uM | ALA1737857 | inconclusive | nM | Homo sapiens | |||
18. | ALA1481784 | SID24827276 | Potency | 4.611 | uM | ALA1737857 | inconclusive | nM | Homo sapiens | |||
19. | ALA1489472 | SID17413966 | Potency | 4.11 | uM | ALA1737857 | inconclusive | nM | Homo sapiens | |||
20. | ALA1601122 | SID24809792 | Potency | 7.308 | uM | ALA1737857 | inconclusive | nM | Homo sapiens |