# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA563480 | 24 | Ki | > | 10 | uM | ALA3802318 | nM | Homo sapiens | |||
2. | ALA3798598 | 2 | Ki | > | 10 | uM | ALA3802318 | nM | Homo sapiens | |||
3. | ALA3793911 | 31b | Ki | > | 50000 | nM | ALA3794960 | nM | Homo sapiens | |||
4. | Grapiprant (CJ-023,423) | GRAPIPRANT | IC50 | = | 11.7 | nM | ALA3795722 | 7.93 | nM | Homo sapiens | ||
5. | 3-[[6-[3-(hydroxymethyl)phenyl]-3-methylpyridine-2-carbonyl]amino]-2,4-dimethylbenzoic acid | 7a | IC50 | = | 2.36 | nM | ALA3795722 | 8.63 | nM | Homo sapiens | ||
6. | ALA3793928 | 3a | IC50 | = | 14.2 | nM | ALA3795722 | 7.85 | nM | Homo sapiens | ||
7. | ALA3792999 | 3b | IC50 | = | 87.9 | nM | ALA3795722 | 7.06 | nM | Homo sapiens | ||
8. | ALA3792709 | 3c | IC50 | = | 19.5 | nM | ALA3795722 | 7.71 | nM | Homo sapiens | ||
9. | ALA3793956 | 4a | IC50 | = | 16.5 | nM | ALA3795722 | 7.78 | nM | Homo sapiens | ||
10. | ALA3793994 | 4b | IC50 | = | 84 | nM | ALA3795722 | 7.08 | nM | Homo sapiens | ||
11. | ALA3793002 | 4c | IC50 | = | 1.61 | nM | ALA3795722 | 8.79 | nM | Homo sapiens | ||
12. | ALA3793924 | 4d | IC50 | = | 39.8 | nM | ALA3795722 | 7.40 | nM | Homo sapiens | ||
13. | ALA3793912 | 4e | IC50 | = | 96.7 | nM | ALA3795722 | 7.01 | nM | Homo sapiens | ||
14. | ALA3686863 | BDBM142234 | IC50 | = | 5.62 | nM | ALA3795722 | 8.25 | nM | Homo sapiens | ||
15. | Grapiprant (CJ-023,423) | GRAPIPRANT | IC50 | = | 1520 | nM | ALA3795721 | 5.82 | nM | Homo sapiens | ||
16. | 3-[[6-[3-(hydroxymethyl)phenyl]-3-methylpyridine-2-carbonyl]amino]-2,4-dimethylbenzoic acid | 7a | IC50 | = | 38.7 | nM | ALA3795721 | 7.41 | nM | Homo sapiens | ||
17. | ALA3793928 | 3a | IC50 | = | 2890 | nM | ALA3795721 | 5.54 | nM | Homo sapiens | ||
18. | ALA3792709 | 3c | IC50 | = | 1450 | nM | ALA3795721 | 5.84 | nM | Homo sapiens | ||
19. | ALA3793956 | 4a | IC50 | = | 1450 | nM | ALA3795721 | 5.84 | nM | Homo sapiens | ||
20. | ALA3793002 | 4c | IC50 | = | 1160 | nM | ALA3795721 | 5.94 | nM | Homo sapiens |