# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA378376 | 16c | Ki | = | 2 | nM | ALA5242762 | 8.70 | nM | Homo sapiens | ||
2. | ALA5272661 | 8; PF-04475270 | Ki | < | 2 | nM | ALA5242762 | nM | Homo sapiens | |||
3. | ALA378376 | 16c | IC50 | = | 2 | nM | ALA5242761 | 8.70 | nM | Homo sapiens | ||
4. | ALA5272661 | 8; PF-04475270 | IC50 | = | 2 | nM | ALA5242761 | 8.70 | nM | Homo sapiens | ||
5. | ALA3286660 | 7z, TG8-15 | Kb | = | 15 | uM | ALA5224044 | nM | Homo sapiens | |||
6. | TG 4-155 | SID17515129 | Kb | = | 11.4 | uM | ALA5224034 | nM | Homo sapiens | |||
7. | ALA5285583 | PF-04852946 (2) | Ki | = | 16.3 | uM | ALA5224030 | 4.79 | nM | Homo sapiens | ||
8. | PF 04418948 | 15, PF-04418948 | Ki | > | 10 | uM | ALA5224027 | nM | Homo sapiens | |||
9. | BAY 876 | 66; BAY-876 | IC50 | = | 1.12 | uM | ALA5214528 | 5.95 | nM | Homo sapiens | ||
10. | BAY-474 | EUB0000293 | % of inhibition | = | 19 | % | ALA5213239 | % | Homo sapiens | |||
11. | 4-[[[2-[(4-fluorophenyl)methyl]-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carbonyl]amino]methyl]benzoic acid | 47 | Activity | 0 | ALA5168437 | Active | Homo sapiens | |||||
12. | 4-[[[2-[(4-fluorophenyl)methyl]-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carbonyl]amino]methyl]benzoic acid | 47 | pA2 | = | 8.173 | ALA5168423 | 8.17 | nM | Homo sapiens | |||
13. | 4-[[[2-[(4-fluorophenyl)methyl]-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carbonyl]amino]methyl]benzoic acid | 47 | IC50 | = | 2.7 | nM | ALA5168422 | 8.57 | nM | Homo sapiens | ||
14. | 4-[[[2-[(4-fluorophenyl)methyl]-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carbonyl]amino]methyl]benzoic acid | 47 | IC50 | = | 5 | nM | ALA5168421 | 8.30 | nM | Homo sapiens | ||
15. | E7046 (ER-886406) | BDBM119448 | IC50 | = | 18.5 | nM | ALA5168421 | 7.73 | nM | Homo sapiens | ||
16. | ALA5184401 | 57 | IC50 | > | 1000 | nM | ALA5168387 | nM | Homo sapiens | |||
17. | ALA5205020 | 51 | IC50 | > | 1000 | nM | ALA5168387 | nM | Homo sapiens | |||
18. | ALA5175609 | 28 | IC50 | > | 1000 | nM | ALA5168387 | nM | Homo sapiens | |||
19. | ALA5185966 | 26 | IC50 | > | 1000 | nM | ALA5168387 | nM | Homo sapiens | |||
20. | ALA5194028 | 24 | IC50 | > | 1000 | nM | ALA5168387 | nM | Homo sapiens |