# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5274986 | (N)-mc Ado | Ki | > | 50000 | nM | ALA5233318 | nM | Homo sapiens | |||
2. | ALA2112095 | 5d | Ki | > | 50000 | nM | ALA5233318 | nM | Homo sapiens | |||
3. | ALA252048 | 28, CVT-6694 | Ki | = | 5.5 | nM | ALA5223708 | 8.26 | nM | Homo sapiens | ||
4. | Caffeine | caffeine | pKi | = | 4.5 | ALA5223690 | 4.50 | nM | Homo sapiens | |||
5. | Caffeine | caffeine | IC50 | = | 10.4 | uM | ALA5223690 | 4.98 | nM | Homo sapiens | ||
6. | Theobromine | theobromine | IC50 | = | 130 | uM | ALA5223690 | nM | Homo sapiens | |||
7. | Caffeine | caffeine | pKi | = | 4.5 | ALA5223685 | 4.50 | nM | Homo sapiens | |||
8. | MRS 1706 | 20 | Ki | = | 1.39 | nM | ALA5223681 | 8.86 | nM | Homo sapiens | ||
9. | MRS 1754 | 27 | Ki | = | 1.97 | nM | ALA5223681 | 8.71 | nM | Homo sapiens | ||
10. | PSB 1115 | 6c (PSB-1115) | Ki | = | 53.4 | nM | ALA5223681 | 7.27 | nM | Homo sapiens | ||
11. | (R)-PFI 2 hydrochloride | EUB0000196bCl | Ki | = | 1.3 | uM | ALA5214692 | 5.89 | nM | Homo sapiens | ||
12. | PF 05105679 | 8, PF-05105679 | % of effect | = | 21 | % | ALA5214511 | % | Homo sapiens | |||
13. | MRK-740 | EUB0000234b | EC50 | > | 10 | uM | ALA5214652 | nM | Homo sapiens | |||
14. | MRK-740 | EUB0000234b | % of inhibition | > | 50 | % | ALA5214651 | % | Homo sapiens | |||
15. | ALA5188801 | 30i | Ki | = | 2495.5 | nM | ALA5164006 | 5.60 | nM | Homo sapiens | ||
16. | ALA5201523 | 30c | Ki | = | 513 | nM | ALA5164006 | 6.29 | nM | Homo sapiens | ||
17. | ALA5199428 | 14c | Ki | > | 10000 | nM | ALA5164006 | nM | Homo sapiens | |||
18. | Imaradenant (AZD4635) | IMARADENANT | Ki | = | 55.8 | nM | ALA5148527 | 7.25 | nM | Homo sapiens | ||
19. | ALA5203105 | 12o 2HCl | Ki | = | 40.6 | nM | ALA5148527 | 7.39 | nM | Homo sapiens | ||
20. | ALA5176737 | 12o | Ki | = | 96.7 | nM | ALA5148527 | 7.01 | nM | Homo sapiens |