# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Sildenafil | 1 | IC50 | = | 3.6 | nM | ALA5246775 | 8.44 | nM | Homo sapiens | ||
2. | 5-(2-Ethoxyphenyl)-1-methyl-3-n-propyl-1,6-dihydro-7H-pyrazolo[4,3-d]-7-pyrimidinone | III | IC50 | = | 27 | nM | ALA5246775 | 7.57 | nM | Homo sapiens | ||
3. | ALA51814 | II | IC50 | = | 330 | nM | ALA5246775 | 6.48 | nM | Homo sapiens | ||
4. | ALA28079 | M&B-22948 | IC50 | = | 2000 | nM | ALA5246775 | 5.70 | nM | Homo sapiens | ||
5. | ALA5289112 | 2-2 | INH | = | 100 | % | ALA5243070 | % | Homo sapiens | |||
6. | ALA5285980 | 2-1 | INH | = | 100 | % | ALA5243070 | % | Homo sapiens | |||
7. | ALA5283454 | 2 | INH | = | 100 | % | ALA5243070 | % | Homo sapiens | |||
8. | ALA2137306 | SID99356275 | INH | = | 100 | % | ALA5235756 | % | Homo sapiens | |||
9. | ALA5281261 | 176 | INH | = | 100 | % | ALA5235756 | % | Homo sapiens | |||
10. | ALA3338445 | 19a, T-6932 | IC50 | = | 0.16 | nM | ALA5235622 | 9.80 | nM | Homo sapiens | ||
11. | ALA4641729 | 8i | Ki | = | 86 | nM | ALA5235563 | 7.07 | nM | Homo sapiens | ||
12. | ALA163905 | 18 | Ki | = | 4 | nM | ALA5235563 | 8.40 | nM | Homo sapiens | ||
13. | ALA349947 | 15b | Ki | = | 63 | nM | ALA5235563 | 7.20 | nM | Homo sapiens | ||
14. | ALA166025 | 12c | Ki | = | 64 | nM | ALA5235563 | 7.19 | nM | Homo sapiens | ||
15. | ALA165117 | 12g | Ki | = | 64 | nM | ALA5235563 | 7.19 | nM | Homo sapiens | ||
16. | ALA349204 | 12i | Ki | = | 64 | nM | ALA5235563 | 7.19 | nM | Homo sapiens | ||
17. | ALA350962 | 12f | Ki | = | 51 | nM | ALA5235563 | 7.29 | nM | Homo sapiens | ||
18. | ALA166018 | 12j | Ki | = | 51 | nM | ALA5235563 | 7.29 | nM | Homo sapiens | ||
19. | ALA133285 | 3 | Ki | = | 9 | nM | ALA5235563 | 8.05 | nM | Homo sapiens | ||
20. | ALA5275513 | 150 | IC50 | = | 126 | nM | ALA5235562 | 6.90 | nM | Homo sapiens |