# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5278465 | 33 | IC50 | > | 50 | uM | ALA5252926 | nM | Homo sapiens | |||
2. | GNF 5837 | 22, GNF-5837 | Delta TM | = | 0.42 | C | ALA5209756 | C | Homo sapiens | |||
3. | GNF 5837 | 22, GNF-5837 | Delta TM | = | 0.28 | C | ALA5209756 | C | Homo sapiens | |||
4. | XL019 | XL019; 3 | Delta TM | = | 0.84 | C | ALA5209756 | C | Homo sapiens | |||
5. | Roscovitine (Seliciclib,CYC202) | Roscovitine | Delta TM | = | 0 | C | ALA5209756 | C | Homo sapiens | |||
6. | ALA5169393 | 11 | INH | = | 66 | % | ALA5157102 | % | Homo sapiens | |||
7. | ALA5182980 | 4 | INH | = | 71 | % | ALA5157102 | % | Homo sapiens | |||
8. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405440 | % | Homo sapiens | |||
9. | ALA4559936 | (+/-)-6 | Activity | = | 46 | % | ALA4391429 | % | Homo sapiens | |||
10. | ALA4564973 | 50 | INH | = | 69 | % | ALA4389803 | % | Homo sapiens | |||
11. | ALA4555459 | 43 | INH | = | 41 | % | ALA4389326 | % | Homo sapiens | |||
12. | ALA4473365 | 7c | Activity | = | 57 | % | ALA4382607 | % | Homo sapiens | |||
13. | ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379296 | nM | Homo sapiens | |||
14. | ALA4459587 | DC-TEADin02 | INH | = | -13 | % | ALA4378898 | % | Homo sapiens | |||
15. | CDK9-IN-7 | 21e | INH | = | 2 | % | ALA4377750 | % | Homo sapiens | |||
16. | ALA4462318 | 19i | Kd(free) | = | 7.086 | uM | ALA4371348 | 5.15 | nM | Homo sapiens | ||
17. | ALA4443828 | 19h | Kd(free) | = | 4.455 | uM | ALA4371348 | 5.35 | nM | Homo sapiens | ||
18. | Dasatinib | 2, BMS-354825 | Activity | > | 75 | % | ALA4807900 | % | Homo sapiens | |||
19. | ALA4855726 | B3 | Activity | > | 75 | % | ALA4807900 | % | Homo sapiens | |||
20. | ALA4867844 | C7 | Activity | > | 75 | % | ALA4807900 | % | Homo sapiens |