# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5306285 | EUB0002235 | delta Tm Staurosporine positive control | = | 8.802 | ALA5304810 | Homo sapiens | |||||
2. | ALA5306285 | EUB0002235 | delta Tm | = | -0.371 | ALA5304810 | Not Active | Homo sapiens | ||||
3. | ALA5308262 | EUB0002234 | delta Tm Staurosporine positive control | = | 8.802 | ALA5304706 | Homo sapiens | |||||
4. | ALA5308262 | EUB0002234 | delta Tm | = | -1.352 | ALA5304706 | Not Active | Homo sapiens | ||||
5. | ALA5308250 | EUB0002186 | delta Tm Staurosporine positive control | = | 7.9 | ALA5304672 | Homo sapiens | |||||
6. | ALA5308250 | EUB0002186 | delta Tm | = | 0.316 | ALA5304672 | Not Active | Homo sapiens | ||||
7. | ALA5306577 | EUB0002354 | delta Tm Staurosporine positive control | = | 7.9 | ALA5304573 | Homo sapiens | |||||
8. | ALA5306577 | EUB0002354 | delta Tm | = | 0.222 | ALA5304573 | Not Active | Homo sapiens | ||||
9. | ALA3774632 | 5b | Activity | = | 79 | % | ALA3777892 | % | Homo sapiens | |||
10. | ALA3774537 | 54k | INH | 0 | ALA3777935 | Not Active | % | Homo sapiens | ||||
11. | ALA3758502 | 1 | INH | = | 4.3 | % | ALA3761273 | % | Homo sapiens | |||
12. | ALA3746293 | 23 | INH | = | 7.2 | % | ALA3751244 | % | Homo sapiens | |||
13. | ALA3703188 | BDBM47183 | IC50 | = | 132 | nM | ALA3705586 | 6.88 | 198712 | nM | Homo sapiens | |
14. | ALA3633152 | 24 | Kd | = | 81 | nM | ALA3635833 | 7.09 | nM | Homo sapiens | ||
15. | ALA3633152 | 24 | Activity | = | 4 | % | ALA3635822 | % | Homo sapiens | |||
16. | AZ 3146 | SID137275933 | IC50 | = | 35 | uM | ALA5253677 | nM | Homo sapiens | |||
17. | CC-671 | 23; CC-671 | IC50 | = | 5 | nM | ALA5237387 | 8.30 | nM | Homo sapiens | ||
18. | ALA4449557 | 10; NTRC 0066-0 | IC50 | = | 0.6 | nM | ALA5227240 | 9.22 | nM | Homo sapiens | ||
19. | Defactinib | DEFACTINIB | % of control | = | 8.3 | % | ALA5213440 | % | Homo sapiens | |||
20. | omipalisib | SID137275909 | % of control | = | 4 | % | ALA5213179 | % | Homo sapiens |