# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | NMS-E973 | 18, NMS-E973 | IC50 | > | 10 | nM | ALA2443992 | nM | Homo sapiens | |||
2. | ALA2443138 | 30 | IC50 | > | 10 | nM | ALA2443992 | nM | Homo sapiens | |||
3. | ALA2443139 | 31 | IC50 | > | 10 | nM | ALA2443992 | nM | Homo sapiens | |||
4. | ALA2443026 | 38 | IC50 | > | 10 | nM | ALA2443992 | nM | Homo sapiens | |||
5. | ALA2425654 | 3 | INH | = | 99 | % | ALA2429296 | % | Homo sapiens | |||
6. | ALA2425652 | 4 | INH | = | 96 | % | ALA2429296 | % | Homo sapiens | |||
7. | ALA2425649 | 8 | INH | = | 98 | % | ALA2429296 | % | Homo sapiens | |||
8. | ALA2425645 | 11 | INH | = | 100 | % | ALA2429296 | % | Homo sapiens | |||
9. | ALA2425644 | 13 | INH | = | 100 | % | ALA2429296 | % | Homo sapiens | |||
10. | ALA2425628 | 24f | Kd | = | 1.9 | uM | ALA2429166 | 5.72 | nM | Homo sapiens | ||
11. | ALA2425628 | 24f | INH | > | 85 | % | ALA2429296 | % | Homo sapiens | |||
12. | ALA2425646 | 12 | INH | = | 84 | % | ALA2429296 | % | Homo sapiens | |||
13. | ALA2402081 | 37 | INH | = | 8 | % | ALA2405485 | % | Homo sapiens | |||
14. | NMS-P715 | 15, NMS-P715 | IC50 | = | 8 | nM | ALA2383389 | 8.10 | nM | Homo sapiens | ||
15. | ALA1725279 | SP-600125 | IC50 | = | 98 | nM | ALA2383389 | 7.01 | nM | Homo sapiens | ||
16. | ALA2380574 | 9a | IC50 | = | 438 | nM | ALA2383388 | 6.36 | nM | Homo sapiens | ||
17. | ALA2380575 | 9b | IC50 | = | 116 | nM | ALA2383388 | 6.94 | nM | Homo sapiens | ||
18. | ALA2380576 | 9c | IC50 | = | 189 | nM | ALA2383388 | 6.72 | nM | Homo sapiens | ||
19. | ALA2380577 | 9d | IC50 | = | 28 | nM | ALA2383388 | 7.55 | nM | Homo sapiens | ||
20. | ALA2380578 | 17a | IC50 | = | 17 | nM | ALA2383388 | 7.77 | nM | Homo sapiens |